SCHEMBL29696199

SCHEMBL29696199

O=[N+]([O-])c1cc(OC(F)(F)F)ccc1Br

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.44
GAA P10253 2/20 0.44
ALDH1A1 P00352 6/20 0.43
CYP2D6 P10635 1/20 0.43
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
MITF O75030 1/20 0.41
TP53 P04637 1/20 0.40
CASP3 P42574 1/20 0.40
HTT P42858 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
SENP7 Q9BQF6 1/20 0.40
THRB P10828 2/20 0.39
POLB P06746 1/20 0.39
GPR3 P46089 1/20 0.39
KDM4E B2RXH2 2/20 0.38
TXNRD1 Q16881 1/20 0.38
LMNA P02545 3/20 0.38
HPGD P15428 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3257088 1.00 MAPT (0.44) MAPTGAAALDH1A1CYP2D6MEN1
SCHEMBL8211036 0.83 ALDH1A1 (0.46) MAPTGAAALDH1A1CYP2D6MEN1
SCHEMBL31237064 0.81 ALDH1A1 (0.53) MAPTGAAALDH1A1MEN1KMT2A
SCHEMBL1275648 0.81 ALDH1A1 (0.53) MAPTGAAALDH1A1MEN1KMT2A
SCHEMBL31191383 0.80 MAPK1 (0.48) MAPTALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL493054 0.80 MAPT (0.44) MAPTGAAALDH1A1CYP2D6MEN1
SCHEMBL3495810 0.80 PARP1 (0.45) MAPTALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL707416 0.80 SMN1; SMN2 (0.51) MAPTALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL31714528 0.80 ALDH1A1 (0.50) MAPTALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL2540815 0.80 ALDH1A1 (0.50) MAPTALDH1A1MEN1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114728910-B Pyrazole derivative for FGFR inhibitor and preparation method thereof 上海奕拓医药科技有限责任公司 2024-05-14 CN disclosed
CN-114728910-A Pyrazole derivatives for FGFR inhibitor and preparation method thereof 上海奕拓医药科技有限责任公司 2022-07-08 CN disclosed