SCHEMBL29699256

SCHEMBL29699256

COC(=O)c1nc(-c2ccc(Cl)cc2Cl)c(C(F)(F)F)cc1N

nearest known ligand 0.66

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CFTR P13569 9/20 0.66
ALPL P05186 1/20 0.43
ABL1 P00519 1/20 0.42
CNR1 P21554 3/20 0.41
MRGPRX4 Q96LA9 1/20 0.41
S1PR4 O95977 1/20 0.40
SLC6A3 Q01959 1/20 0.40
HSP90AB1 P08238 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2371919 1.00 CFTR (0.66) CFTRALPLABL1CNR1MRGPRX4
SCHEMBL23671475 0.94 CFTR (0.59) CFTRALPLABL1CNR1MRGPRX4
SCHEMBL2372275 0.90 CFTR (0.57) CFTRABL1MRGPRX4S1PR4
SCHEMBL29699295 0.90 CFTR (0.57) CFTRABL1MRGPRX4S1PR4
SCHEMBL2371637 0.86 CFTR (0.64) CFTRALPLCNR1HSP90AB1
SCHEMBL29699354 0.86 CFTR (0.64) CFTRALPLCNR1HSP90AB1
SCHEMBL27990279 0.80 CFTR (0.55) CFTRCNR1HSP90AB1
SCHEMBL29798093 0.79 CFTR (1.00) CFTR
SCHEMBL2372654 0.79 CFTR (1.00) CFTR
SCHEMBL29699242 0.79 CFTR (1.00) CFTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3980121-A1 PYRIDINE AND PYRAZINE DERIVATIVE FOR THE TREATMENT OF CF, COPD, AND BRONCHIECTASIS Novartis AG (CH) 2022-04-13 EP disclosed