SCHEMBL29699764

SCHEMBL29699764

COc1ccc(NC(=O)c2cc(C)n(Cc3cccc(N4CCN(C(=O)C5CC5)CC4)c3)n2)cc1

nearest known ligand 0.83

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.83
CYP2C9 P11712 2/20 0.83
MAPT P10636 6/20 0.47
THRB P10828 1/20 0.47
KMT2A Q03164 2/20 0.46
HSD17B10 Q99714 2/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
MTNR1B P49286 1/20 0.46
MEN1 O00255 1/20 0.45
TP53 P04637 1/20 0.45
KDM4E B2RXH2 1/20 0.44
LMNA P02545 3/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
GAA P10253 1/20 0.44
ALDH1A1 P00352 1/20 0.43
MAPK1 P28482 1/20 0.43
AURKA O14965 1/20 0.43
RPS6KB1 P23443 1/20 0.43
PTGER1 P34995 2/20 0.42
DGAT1 O75907 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29699835 0.92 CYP3A4 (0.83) CYP3A4CYP2C9MAPTKMT2AMEN1
SCHEMBL29699818 0.91 CYP3A4 (0.82) CYP3A4CYP2C9MAPTKMT2AMEN1
SCHEMBL29699861 0.91 CYP3A4 (1.00) CYP3A4CYP2C9KMT2AMEN1TP53
SCHEMBL29699844 0.88 CYP3A4 (1.00) CYP3A4CYP2C9MAPTKMT2AMEN1
SCHEMBL29699913 0.86 CYP3A4 (0.75) CYP3A4CYP2C9MAPTKMT2AMEN1
SCHEMBL29700058 0.81 CYP3A4 (0.83) CYP3A4CYP2C9MAPTKMT2AL3MBTL1
SCHEMBL29699900 0.79 CYP3A4 (0.81) CYP3A4CYP2C9KMT2AMEN1TP53
SCHEMBL29699779 0.78 MEN1 (0.64) CYP3A4CYP2C9MAPTKMT2AHSD17B10
SCHEMBL29699929 0.76 CYP3A4 (0.76) CYP3A4CYP2C9MAPTKMT2AMEN1
SCHEMBL29699716 0.76 CYP3A4 (0.76) CYP3A4CYP2C9MAPTKMT2AHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114685371-A Pyrazole carboxamide derivatives, their preparation and use 四川大学 2022-07-01 CN claimed
CN-114685371-A Pyrazole carboxamide derivatives, their preparation and use 四川大学 2022-07-01 CN disclosed