SCHEMBL29699861

SCHEMBL29699861

Cc1cc(C(=O)Nc2ccc(OC(F)(F)F)cc2)nn1Cc1cccc(N2CCN(C(=O)C3CC3)CC2)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 1.00
CYP2C9 P11712 2/20 1.00
SMN1; SMN2 Q16637 1/20 0.47
MCHR1 Q99705 2/20 0.46
EPHX2 P34913 2/20 0.45
TP53 P04637 2/20 0.44
ABL1 P00519 2/20 0.44
KCNH2 Q12809 1/20 0.44
CHRM4 P08173 4/20 0.44
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
NPY5R Q15761 1/20 0.43
PTGER1 P34995 1/20 0.41
GCGR P47871 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29699764 0.91 CYP3A4 (0.83) CYP3A4CYP2C9SMN1; SMN2TP53MEN1
SCHEMBL29700058 0.91 CYP3A4 (0.83) CYP3A4CYP2C9SMN1; SMN2EPHX2TP53
SCHEMBL29699844 0.90 CYP3A4 (1.00) CYP3A4CYP2C9EPHX2MEN1KMT2A
SCHEMBL29699900 0.89 CYP3A4 (0.81) CYP3A4CYP2C9SMN1; SMN2TP53ABL1
SCHEMBL29699835 0.89 CYP3A4 (0.83) CYP3A4CYP2C9TP53MEN1KMT2A
SCHEMBL29699818 0.88 CYP3A4 (0.82) CYP3A4CYP2C9TP53MEN1KMT2A
SCHEMBL29699929 0.87 CYP3A4 (0.76) CYP3A4CYP2C9SMN1; SMN2TP53ABL1
SCHEMBL29699910 0.86 CYP3A4 (0.76) CYP3A4CYP2C9SMN1; SMN2TP53ABL1
SCHEMBL29699716 0.86 CYP3A4 (0.76) CYP3A4CYP2C9SMN1; SMN2EPHX2TP53
SCHEMBL29699913 0.83 CYP3A4 (0.75) CYP3A4CYP2C9SMN1; SMN2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114685371-A Pyrazole carboxamide derivatives, their preparation and use 四川大学 2022-07-01 CN claimed
CN-114685371-A Pyrazole carboxamide derivatives, their preparation and use 四川大学 2022-07-01 CN disclosed