SCHEMBL29699885

SCHEMBL29699885

O=C(Nc1ccc(OC(F)(F)F)cc1)c1ccn(Cc2cccc(Br)c2)n1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.52
CACNA1G O43497 2/20 0.52
CACNA1H O95180 2/20 0.52
CACNA1I Q9P0X4 2/20 0.52
ABL1 P00519 3/20 0.49
SMN1; SMN2 Q16637 3/20 0.49
KCNH2 Q12809 1/20 0.49
CYP3A4 P08684 1/20 0.46
CYP2C9 P11712 1/20 0.46
HIF1A Q16665 2/20 0.46
HTT P42858 1/20 0.45
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
KDM4E B2RXH2 1/20 0.45
GAA P10253 1/20 0.45
MAPT P10636 1/20 0.45
EPHX2 P34913 1/20 0.45
PPARA Q07869 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.44
HDAC1 Q13547 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15504901 0.85 SMN1; SMN2 (0.52) TP53ABL1SMN1; SMN2KCNH2CYP3A4
SCHEMBL29699842 0.83 CYP3A4 (0.65) TP53ABL1SMN1; SMN2KCNH2CYP3A4
SCHEMBL29699941 0.81 TP53 (0.47) TP53CACNA1GCACNA1HCACNA1IABL1
SCHEMBL29699853 0.80 TP53 (0.50) TP53CACNA1GCACNA1HCACNA1IABL1
SCHEMBL29699805 0.78 CYP3A4 (0.58) TP53CACNA1GCACNA1HCACNA1IABL1
SCHEMBL15504917 0.78 MAPT (0.65) TP53ABL1SMN1; SMN2KCNH2CYP2C9
SCHEMBL31598793 0.74 CACNA1G (0.50) CACNA1GCACNA1HCACNA1IHDAC1SCD
SCHEMBL15504915 0.74 ABL1 (0.47) TP53ABL1SMN1; SMN2KCNH2CYP3A4
SCHEMBL15391824 0.74 ABL1 (0.63) TP53ABL1SMN1; SMN2KCNH2HTT
SCHEMBL29700080 0.73 PTGER1 (0.60) CACNA1GCACNA1ISMN1; SMN2HTTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114685371-A Pyrazole carboxamide derivatives, their preparation and use 四川大学 2022-07-01 CN disclosed