SCHEMBL29701366

SCHEMBL29701366

COc1ccc([C@H](CC(=O)O)NC(=O)C2CC(CCc3ccc4c(n3)NCCC4)C2)cn1

nearest known ligand 0.62

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 20/20 0.62
ITGAV P06756 20/20 0.62
ITGB5 P18084 6/20 0.59
ITGA2B P08514 5/20 0.59
ITGB6 P18564 9/20 0.56
ITGB1 P05556 2/20 0.56
ITGA5 P08648 2/20 0.56
ITGB8 P26012 5/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20140807 1.00 ITGB3 (0.62) ITGB3ITGAVITGB5ITGA2BITGB6
SCHEMBL20140803 1.00 ITGB3 (0.62) ITGB3ITGAVITGB5ITGA2BITGB6
SCHEMBL21317545 1.00 ITGB3 (0.62) ITGB3ITGAVITGB5ITGA2BITGB6
SCHEMBL20158050 1.00 ITGB3 (0.62) ITGB3ITGAVITGB5ITGA2BITGB6
SCHEMBL20158219 0.94 ITGB3 (0.61) ITGB3ITGAVITGB5ITGA2BITGB6
SCHEMBL20142087 0.92 ITGB3 (0.58) ITGB3ITGAVITGB5ITGA2BITGB6
SCHEMBL20142092 0.92 ITGB3 (0.58) ITGB3ITGAVITGB5ITGA2BITGB6
SCHEMBL29701353 0.92 ITGB3 (0.58) ITGB3ITGAVITGB5ITGA2BITGB6
SCHEMBL21314351 0.91 ITGAV (0.61) ITGB3ITGAVITGB5ITGA2BITGB6
SCHEMBL21317480 0.91 ITGAV (0.61) ITGB3ITGAVITGB5ITGA2BITGB6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110167934-B Cyclobutane-and azetidine-containing monocyclic and spiro compounds as alpha V integrin inhibitors 百时美施贵宝公司 2022-06-10 CN claimed