SCHEMBL29702152

SCHEMBL29702152

COc1ccc(C(CC(=O)OC(C)(C)C)C2CC(CCC=Cc3ccc4c(n3)NCCC4)C2)cn1

nearest known ligand 0.47

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ITGAV P06756 20/20 0.47
ITGB3 P05106 18/20 0.47
ITGA2B P08514 3/20 0.43
ITGB5 P18084 1/20 0.43
ITGB6 P18564 6/20 0.43
ITGB1 P05556 2/20 0.41
ITGA5 P08648 2/20 0.41
ITGB8 P26012 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30487505 1.00 ITGAV (0.47) ITGAVITGB3ITGA2BITGB5ITGB6
SCHEMBL20158103 1.00 ITGAV (0.47) ITGAVITGB3ITGA2BITGB5ITGB6
SCHEMBL20141446 0.91 ITGAV (0.54) ITGAVITGB3ITGA2BITGB5ITGB6
SCHEMBL20141445 0.91 ITGAV (0.54) ITGAVITGB3ITGA2BITGB5ITGB6
SCHEMBL20158101 0.85 ITGAV (0.60) ITGAVITGB3ITGA2BITGB5ITGB6
SCHEMBL30487535 0.85 ITGAV (0.60) ITGAVITGB3ITGA2BITGB5ITGB6
SCHEMBL20158099 0.80 CHRNA7 (0.37) ITGAVITGB3ITGA2BITGB5ITGB1
SCHEMBL30487514 0.80 CHRNA7 (0.37) ITGAVITGB3ITGA2BITGB5ITGB1
SCHEMBL21317544 0.79 CHRNA7 (0.36) ITGAVITGB3
SCHEMBL20141277 0.76 ITGAV (0.70) ITGAVITGB3ITGA2BITGB5ITGB6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110167934-B Cyclobutane-and azetidine-containing monocyclic and spiro compounds as alpha V integrin inhibitors 百时美施贵宝公司 2022-06-10 CN disclosed