SCHEMBL29705175

SCHEMBL29705175

CCOC(=O)c1cn(N(CC(F)(F)F)C(=O)OC(C)(C)C)c2ncc(Br)cc2c1=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.43
FOS P01100 2/20 0.36
JUN P05412 2/20 0.36
NFKB1 P19838 2/20 0.36
NFKB2 Q00653 2/20 0.36
RELA Q04206 2/20 0.36
KDM4E B2RXH2 5/20 0.36
GABRA1 P14867 1/20 0.36
GABRB1 P18505 1/20 0.36
GABRA3 P34903 1/20 0.36
GABRB2 P47870 1/20 0.36
ALDH1A1 P00352 4/20 0.35
HSD17B10 Q99714 3/20 0.35
HPGD P15428 2/20 0.35
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
MAPT P10636 3/20 0.35
TSHR P16473 1/20 0.35
MAPK1 P28482 1/20 0.34
GAA P10253 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20521062 1.00 LMNA (0.43) LMNAFOSJUNNFKB1NFKB2
SCHEMBL28735837 0.89 LMNA (0.33) LMNAKDM4EALDH1A1HSD17B10HPGD
SCHEMBL20521561 0.88 KDM4E (0.35) LMNAFOSJUNNFKB1NFKB2
SCHEMBL29705123 0.88 KDM4E (0.35) LMNAFOSJUNNFKB1NFKB2
SCHEMBL20520911 0.88 LMNA (0.41) LMNAFOSJUNNFKB1NFKB2
SCHEMBL23646765 0.86 LMNA (0.44) LMNAFOSJUNNFKB1NFKB2
SCHEMBL3289956 0.80 LMNA (0.50) LMNAKDM4EGABRA1GABRB1GABRA3
SCHEMBL20520865 0.79 PDE4B (0.47) LMNAKDM4EGABRA1GABRB1GABRA3
SCHEMBL20240770 0.78 LMNA (0.46) LMNAKDM4EGABRA1GABRB1GABRA3
SCHEMBL20520759 0.77 GSK3B (0.31) LMNAKDM4EALDH1A1HSD17B10HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110475777-B Novel pyrido [2,3-b ] indole compounds for the treatment and prevention of bacterial infections 豪夫迈·罗氏有限公司 2022-04-15 CN disclosed