SCHEMBL29709458

SCHEMBL29709458

CC(C)(C)OC(=O)N1CCC[C@@H](n2cnc3ccccc3c2=O)C1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR1 Q9BXC0 1/20 0.55
BTK Q06187 4/20 0.49
OPRM1 P35372 3/20 0.45
OGFRL1 Q5TC84 3/20 0.45
OPRD1 P41143 2/20 0.45
OPRK1 P41145 2/20 0.45
EGFR P00533 1/20 0.44
SRC P12931 1/20 0.44
HPGDS O60760 1/20 0.44
JAK2 O60674 1/20 0.43
JAK1 P23458 1/20 0.43
USP30 Q70CQ3 2/20 0.43
PIK3CD O00329 1/20 0.42
PIK3R2 O00459 1/20 0.42
PIK3CA P42336 1/20 0.42
PIK3CB P42338 1/20 0.42
PIK3CG P48736 1/20 0.42
PIK3R5 Q8WYR1 1/20 0.42
PIK3R3 Q92569 1/20 0.42
FPR2 P25090 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16337414 1.00 HCAR1 (0.55) HCAR1BTKOPRM1OGFRL1OPRD1
SCHEMBL16335107 1.00 HCAR1 (0.55) HCAR1BTKOPRM1OGFRL1OPRD1
SCHEMBL19118890 0.86 HCAR1 (0.52) HCAR1EGFRSRCHPGDSJAK2
SCHEMBL19118889 0.86 HCAR1 (0.52) HCAR1EGFRSRCHPGDSJAK2
SCHEMBL16336882 0.86 HCAR1 (0.54) HCAR1BTKHPGDSJAK2JAK1
SCHEMBL16333786 0.86 HCAR1 (0.54) HCAR1BTKHPGDSJAK2JAK1
SCHEMBL19118355 0.84 HCAR1 (0.49) HCAR1JAK2JAK1FPR2MAPT
SCHEMBL19118356 0.84 HCAR1 (0.49) HCAR1JAK2JAK1FPR2MAPT
SCHEMBL16333958 0.84 BTK (0.54) BTKJAK2JAK1ACVR1MAPT
SCHEMBL31032266 0.79 HCAR1 (0.49) HCAR1EGFRSRCHPGDSJAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4008328-A1 PRIMARY CARBOXAMIDES AS BTK INHIBITORS AbbVie Inc. (US) 2022-06-08 EP disclosed