SCHEMBL29709488

SCHEMBL29709488

Cc1c(B2OC(C)(C)C(C)(C)O2)cccc1N1Cc2ccc(F)cc2C1=O

nearest known ligand 0.49

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
BTK Q06187 8/20 0.49
JAK2 O60674 3/20 0.46
PDCD1 Q15116 2/20 0.39
CD274 Q9NZQ7 2/20 0.39
IDO1 P14902 1/20 0.37
TDO2 P48775 1/20 0.37
P2RX7 Q99572 8/20 0.37
ADAM17 P78536 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL144722 1.00 BTK (0.49) BTKJAK2PDCD1CD274IDO1
SCHEMBL148493 0.92 BTK (0.46) BTKJAK2PDCD1CD274IDO1
SCHEMBL147175 0.89 BTK (0.45) BTKJAK2PDCD1CD274
SCHEMBL123338 0.87 BTK (0.46) BTKJAK2PDCD1CD274ADAM17
SCHEMBL17425876 0.86 BTK (0.47) BTKJAK2PDCD1CD274P2RX7
SCHEMBL148927 0.85 NPC1 (0.45) BTKJAK2PDCD1CD274
SCHEMBL15284621 0.85 BTK (0.42) BTKJAK2PDCD1CD274
SCHEMBL151946 0.83 BTK (0.43) BTKJAK2PDCD1CD274
SCHEMBL123774 0.81 BTK (0.46) BTKJAK2PDCD1CD274
SCHEMBL148828 0.80 JAK2 (0.49) BTKJAK2PDCD1CD274IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4008328-A1 PRIMARY CARBOXAMIDES AS BTK INHIBITORS AbbVie Inc. (US) 2022-06-08 EP disclosed