SCHEMBL29709652

SCHEMBL29709652

CC(C)(C)OC(=O)N1CCC2(CC1)CCN(c1ccc(N)c(O)c1)CC2

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.48
LMNA P02545 1/20 0.48
MAPT P10636 1/20 0.48
HDAC2 Q92769 2/20 0.48
HDAC1 Q13547 1/20 0.48
CYP3A4 P08684 4/20 0.46
MAPK1 P28482 2/20 0.46
MEN1 O00255 1/20 0.46
CYP2C19 P33261 1/20 0.46
KMT2A Q03164 1/20 0.46
SMARCA2 P51531 1/20 0.46
SMARCA4 P51532 1/20 0.46
PBRM1 Q86U86 1/20 0.46
GPR119 Q8TDV5 9/20 0.46
USP2 O75604 2/20 0.46
HSD17B10 Q99714 2/20 0.46
PDK2 Q15119 1/20 0.45
HIF1A Q16665 1/20 0.44
CYP11B2 P19099 1/20 0.43
TP53 P04637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24793978 1.00 ALDH1A1 (0.48) ALDH1A1LMNAMAPTHDAC2HDAC1
SCHEMBL29709632 0.92 HDAC2 (0.52) ALDH1A1LMNAMAPTHDAC2HDAC1
SCHEMBL24793976 0.92 HDAC2 (0.52) ALDH1A1LMNAMAPTHDAC2HDAC1
SCHEMBL24793977 0.92 HDAC2 (0.49) ALDH1A1LMNAMAPTHDAC2HDAC1
SCHEMBL29709716 0.92 HDAC2 (0.49) ALDH1A1LMNAMAPTHDAC2HDAC1
SCHEMBL4722818 0.89 MAPT (0.60) ALDH1A1LMNAMAPTMEN1CYP2C19
SCHEMBL31091690 0.87 HDAC2 (0.52) ALDH1A1LMNAMAPTHDAC2HDAC1
SCHEMBL30497506 0.86 CYP3A4 (0.47) ALDH1A1LMNAMAPTHDAC2HDAC1
SCHEMBL17411226 0.86 CYP3A4 (0.47) ALDH1A1LMNAMAPTHDAC2HDAC1
SCHEMBL21946732 0.84 MAPK1 (0.54) ALDH1A1LMNAMAPTCYP3A4MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4581025-A1 PYRIDAZINON DERIVATIVES AS KAT2 DEGRADERS FOR THE TREATMENT OF PROLIFERATIVE DISORDERS Auron Therapeutics, Inc. (US) 2025-07-09 EP disclosed
WO-2024050078-A1 PYRIDAZINON DERIVATIVES AS KAT2 DEGRADERS FOR THE TREATMENT OF PROLIFERATIVE DISORDERS AURON THERAPEUTICS, INC. (US) 2024-03-07 WO disclosed
US-20220402901-A1 SUBSTITUTED N-HETEROCYCLIC CARBOXAMIDES AS ACID CERAMIDASE INHIBITORS AND THEIR USE AS MEDICAMENTS BIAL R&D INVEST S A (PT) 2022-12-22 US disclosed
EP-4031535-A1 SUBSTITUTED N-HETEROCYCLIC CARBOXAMIDES AS ACID CERAMIDASE INHIBITORS AND THEIR USE AS MEDICAMENTS Bial-R&D Investments, S.A. (PT) 2022-07-27 EP disclosed
CN-114761386-A Substituted N-heterocyclic carboxamides as acid ceramidase inhibitors and their use as pharmaceuticals 比亚尔R&D投资股份公司 2022-07-15 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220402901-A1 SUBSTITUTED N-HETEROCYCLIC CARBOXAMIDES AS ACID CERAMIDASE INHIBITORS AND THEIR USE AS MEDICAMENTS ASAH2, ASAH1, GBA1 ALDH1A1 1191/4885LMNA 828/4885MAPT 1369/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.