SCHEMBL29709869

SCHEMBL29709869

O=C(Nc1cccnc1)C1CC(=O)N(c2ccccc2)C1

nearest known ligand 0.81

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.69
CA12 O43570 2/20 0.60
CA1 P00915 2/20 0.60
CA4 P22748 2/20 0.60
CA6 P23280 2/20 0.60
CA7 P43166 2/20 0.60
CA13 Q8N1Q1 2/20 0.60
CA2 P00918 1/20 0.60
CA9 Q16790 1/20 0.60
CA5B Q9Y2D0 1/20 0.60
ALDH1A1 P00352 1/20 0.60
POLB P06746 2/20 0.60
MAPT P10636 1/20 0.59
TDP1 Q9NUW8 1/20 0.59
GAA P10253 1/20 0.56
ROCK2 O75116 1/20 0.56
ROCK1 Q13464 1/20 0.56
MEN1 O00255 1/20 0.56
L3MBTL1 Q9Y468 1/20 0.56
SMN1; SMN2 Q16637 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5843116 0.83 CA12 (0.72) KMT2ACA12CA1CA4CA6
SCHEMBL5841502 0.81 POLB (0.72) KMT2ACA12CA1CA4CA6
SCHEMBL12245738 0.78 KMT2A (0.59) KMT2ACA12CA1CA4CA6
SCHEMBL21150842 0.77 CA12 (0.68) KMT2ACA12CA1CA4CA6
SCHEMBL5842380 0.77 CA12 (0.68) KMT2ACA12CA1CA4CA6
SCHEMBL5843350 0.76 MAPT (0.72) KMT2ACA12CA1CA4CA6
SCHEMBL5842225 0.76 ALDH1A1 (0.77) KMT2ACA12CA1CA4CA6
SCHEMBL2380600 0.76 TSHR (0.52) KMT2ACA12CA1CA4CA6
SCHEMBL12728561 0.75 ALDH1A1 (0.62) KMT2ACA12CA1CA4CA6
SCHEMBL5841136 0.75 TP53 (0.68) CA12CA1CA4CA6CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4003009-A1 SECOND GENERATION INHIBITORS OF MITOCHONDRIAL PERMEABILITY TRANSITION PORE WITH IMPROVED PLASMA STABILITY Oregon Health & Science University (US) 2022-06-01 EP disclosed