SCHEMBL29720900

SCHEMBL29720900

CC(C)n1cc(C(N)=O)c(=O)c(-c2ccc(F)cc2)c1C(N)=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 7/20 0.42
TGFBR2 P37173 5/20 0.42
TNIK Q9UKE5 1/20 0.38
ADORA2A P29274 1/20 0.38
ADORA1 P30542 1/20 0.38
HMGCR P04035 1/20 0.37
PTGDR2 Q9Y5Y4 1/20 0.35
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA9 Q16790 1/20 0.34
IKBKB O14920 2/20 0.33
MEN1 O00255 1/20 0.33
JAK2 O60674 1/20 0.33
EIF2AK2 P19525 1/20 0.33
KMT2A Q03164 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
ELANE P08246 1/20 0.33
RET P07949 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29720980 0.89 TGFBR1 (0.39) TGFBR1TGFBR2TNIKADORA2AADORA1
SCHEMBL29720962 0.89 TGFBR1 (0.39) TGFBR1TGFBR2TNIKADORA2AADORA1
SCHEMBL29811072 0.87 ELANE (0.43) TGFBR1TGFBR2HMGCRPTGDR2ELANE
Hydrochloric Acid SCHEMBL29812369 0.86 ELANE (0.42) TGFBR1TGFBR2HMGCRPTGDR2ELANE
SCHEMBL29720973 0.84 TGFBR1 (0.40) TGFBR1TGFBR2TNIKADORA2AADORA1
SCHEMBL28346481 0.82 MAP2K1 (0.40) TGFBR1TGFBR2CA12CA1CA2
SCHEMBL29720714 0.76 MEN1 (0.44) TGFBR1TGFBR2CA12CA1CA2
SCHEMBL21776525 0.75 SMN1; SMN2 (0.41) PTGDR2MEN1KMT2A
SCHEMBL22188195 0.75 ELANE (0.43) HMGCRPTGDR2ELANE
SCHEMBL29720960 0.74 MEN1 (0.48) TGFBR1TGFBR2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110627796-B Nitrogenous heterocyclic derivative and application thereof in medicine 北京越之康泰生物医药科技有限公司 2022-07-12 CN disclosed