SCHEMBL29754255

SCHEMBL29754255

O=C(O)Cc1ccc(Br)cc1C(F)(F)F

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
RXRA P19793 5/20 0.46
RXRB P28702 5/20 0.46
RXRG P48443 5/20 0.46
POLQ O75417 8/20 0.43
PTGDR2 Q9Y5Y4 1/20 0.42
PTGS2 P35354 2/20 0.40
KDM1A O60341 2/20 0.38
EPRS1 P07814 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20563511 1.00 RXRA (0.46) RXRARXRBRXRGPOLQPTGDR2
SCHEMBL6717126 0.85 KDM1A (0.41) RXRARXRBRXRGPOLQKDM1A
SCHEMBL22235493 0.85 POLQ (0.42) RXRARXRBRXRGPOLQPTGDR2
SCHEMBL15532197 0.83 FFAR4 (0.45) RXRARXRBRXRGPTGDR2
SCHEMBL20562983 0.81 NOTUM (0.43) POLQPTGDR2
SCHEMBL30716953 0.81 POLQ (0.61) RXRARXRBRXRGPOLQPTGDR2
SCHEMBL3741058 0.81 POLQ (0.61) RXRARXRBRXRGPOLQPTGDR2
SCHEMBL892786 0.81 IDO1 (0.53) RXRARXRBRXRGPOLQPTGDR2
SCHEMBL14793818 0.81 CAMK2A (0.47) RXRARXRBRXRGPOLQPTGS2
SCHEMBL29009933 0.80 PTGDR2 (0.37) RXRARXRBRXRGPOLQPTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114436955-B Tetrahydroquinoline and benzomorpholine derivatives or salts thereof, and preparation method and application thereof 复旦大学 2024-08-09 CN disclosed
CN-111032647-B Lysophosphatidic acid receptor 1 (LPAR 1) inhibitor compounds 伊莱利利公司 2023-05-02 CN disclosed
CN-114436955-A Tetrahydroquinoline and benzomorpholine derivatives or salts thereof, and preparation method and application thereof 复旦大学 2022-05-06 CN disclosed