SCHEMBL29759299

SCHEMBL29759299

COc1ccc(F)cc1-c1cc(F)cc(C(=O)NC[C@@H](NC(=O)OCc2ccccc2)C(=O)O)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGER1 P34995 1/20 0.42
MAPT P10636 3/20 0.41
LMNA P02545 1/20 0.41
ITGA4 P13612 1/20 0.41
ITGB7 P26010 1/20 0.41
ITGAV P06756 7/20 0.41
ITGB3 P05106 6/20 0.41
ITGA2B P08514 2/20 0.41
EGLN2 Q96KS0 1/20 0.40
EGLN1 Q9GZT9 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
AAK1 Q2M2I8 1/20 0.40
CYP3A4 P08684 4/20 0.40
ALDH1A1 P00352 3/20 0.40
TP53 P04637 1/20 0.40
KCNH2 Q12809 1/20 0.40
KYNU Q16719 1/20 0.39
TSHR P16473 1/20 0.39
CASP1 P29466 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29759255 0.95 PTGER1 (0.42) PTGER1MAPTLMNAMEN1KMT2A
SCHEMBL29759249 0.90 PTGER1 (0.46) PTGER1MAPTLMNAAAK1CYP3A4
SCHEMBL29759264 0.87 ITGB3 (0.41) PTGER1ITGAVITGB3ITGA2BEGLN2
SCHEMBL29759284 0.82 PTGER1 (0.41) PTGER1MAPTLMNACYP3A4ALDH1A1
SCHEMBL29759270 0.81 ITGB3 (0.37) PTGER1ITGAVITGB3ITGA2BEGLN2
SCHEMBL24526778 0.79 CTSA (0.44) KCNH2
SCHEMBL29759089 0.79 CTSA (0.44) KCNH2
SCHEMBL29759256 0.77 ITGB3 (0.41) PTGER1ITGAVITGB3ITGA2BCASP1
SCHEMBL24527117 0.76 LRRK2 (0.46) ALDH1A1KCNH2
SCHEMBL29742520 0.75 CYP3A4 (0.46) CYP3A4ALDH1A1KYNUTSHRCASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022129047-A2 NOVEL MODULATORS OF THE NMDA RECEPTOR H. LUNDBECK A/S (DK) 2022-06-23 WO disclosed