SCHEMBL29763036

SCHEMBL29763036

O=C(O)N1CCN(c2ccc(S(=O)(=O)N3CCC(Nc4ncc(C(F)(F)F)c(O[C@H]5CCOC5)n4)CC3)cc2)CC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AXL P30530 4/20 0.43
MERTK Q12866 4/20 0.43
TYRO3 Q06418 3/20 0.43
CDK2 P24941 3/20 0.42
CDK1 P06493 2/20 0.42
CCNB1 P14635 2/20 0.42
CCNE1 P24864 2/20 0.42
CCR6 P51684 3/20 0.41
TRPV1 Q8NER1 1/20 0.41
IKBKB O14920 3/20 0.41
CHUK O15111 1/20 0.41
MAPK8 P45983 1/20 0.41
MAPK9 P45984 1/20 0.41
MAPK10 P53779 1/20 0.41
MAPK11 Q15759 1/20 0.41
MAPK14 Q16539 1/20 0.41
KDR P35968 1/20 0.39
CCNT1 O60563 1/20 0.39
CDK4 P11802 1/20 0.39
CCND1 P24385 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26919164 1.00 AXL (0.43) AXLMERTKTYRO3CDK2CDK1
SCHEMBL26919173 1.00 AXL (0.43) AXLMERTKTYRO3CDK2CDK1
SCHEMBL26944092 0.91 IKBKB (0.47) AXLMERTKTYRO3CDK2CDK1
SCHEMBL30697116 0.91 MERTK (0.44) AXLMERTKTYRO3CDK2CDK1
SCHEMBL26943302 0.90 IKBKB (0.45) AXLMERTKTYRO3CDK2CDK1
SCHEMBL26943178 0.88 CDK2 (0.44) AXLMERTKTYRO3CDK2CDK1
SCHEMBL26943177 0.88 CDK2 (0.43) AXLMERTKTYRO3CDK2CDK1
SCHEMBL26943237 0.88 MERTK (0.44) AXLMERTKTYRO3CDK2CDK1
SCHEMBL26943284 0.88 CDK2 (0.41) AXLMERTKTYRO3CDK2CDK1
SCHEMBL29763020 0.87 CCR6 (0.42) AXLMERTKTYRO3CDK2CDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022166793-A1 CDK INHIBITOR 上海齐鲁制药研究中心有限公司 2022-08-11 WO disclosed