SCHEMBL29763402

SCHEMBL29763402

CC(C)COC(=O)Nc1nc(Nc2ccccc2)nc(-c2ccccc2)n1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
IDH2 P48735 1/20 0.49
ALDH1A1 P00352 3/20 0.48
LMNA P02545 2/20 0.48
KDM4E B2RXH2 1/20 0.43
CSNK2A2 P19784 1/20 0.43
CSNK2A1 P68400 1/20 0.43
HPGD P15428 1/20 0.43
KCNH3 Q9ULD8 1/20 0.43
RHOA P61586 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
HSD17B10 Q99714 1/20 0.42
MAOB P27338 1/20 0.41
RORC P51449 2/20 0.41
ADORA1 P30542 2/20 0.41
ADORA3 P0DMS8 1/20 0.41
ADORA2A P29274 1/20 0.41
GLS O94925 1/20 0.41
HTT P42858 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15102521 1.00 IDH2 (0.49) IDH2ALDH1A1LMNAKDM4ECSNK2A2
SCHEMBL27987836 0.88 IDH2 (0.47) IDH2ALDH1A1LMNAHPGDKCNH3
SCHEMBL15102519 0.86 LMNA (0.54) IDH2ALDH1A1LMNAKDM4EHPGD
SCHEMBL16392087 0.85 MEN1 (0.52) ALDH1A1LMNAKDM4ECSNK2A2CSNK2A1
SCHEMBL15102348 0.84 IDH2 (0.52) IDH2ALDH1A1LMNAHPGDKCNH3
SCHEMBL15102561 0.83 IDH2 (0.55) IDH2ALDH1A1LMNAHPGDRHOA
SCHEMBL15102371 0.80 PTGIR (0.52) IDH2ALDH1A1RHOASMN1; SMN2MAOB
SCHEMBL15102360 0.80 ADORA1 (0.59) IDH2ALDH1A1LMNAHPGDKCNH3
SCHEMBL15094826 0.79 IDH2 (0.59) IDH2ALDH1A1LMNARHOARORC
SCHEMBL15102281 0.79 IDH2 (0.55) IDH2ALDH1A1LMNAKDM4EKCNH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115536635-A Therapeutically active compounds and methods of use thereof 法国施维雅药厂 2022-12-30 CN disclosed
CN-115521264-A Therapeutically active compounds and methods of use thereof 法国施维雅药厂 2022-12-27 CN disclosed
CN-114933585-A Therapeutically active compounds and methods of use thereof 法国施维雅药厂 2022-08-23 CN disclosed
CN-108912066-B Therapeutically active compounds and methods of use thereof 安吉奥斯医药品有限公司 2022-06-24 CN disclosed