SCHEMBL29763525

SCHEMBL29763525

COc1ccc(B2OC(C)(C)C(C)(C)O2)c2cc(C(C)(C)C)[nH]c12

nearest known ligand 0.35

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.35
KDM4E B2RXH2 1/20 0.35
EGFR P00533 3/20 0.33
CSF1R P07333 1/20 0.33
NQO2 P16083 2/20 0.31
ALDH1A1 P00352 1/20 0.31
CYP19A1 P11511 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12755285 0.79 KDM4E (0.51) HPGDKDM4ENQO2ALDH1A1CYP19A1
SCHEMBL15186918 0.76 EGFR (0.33) HPGDKDM4EEGFRCSF1R
SCHEMBL20577550 0.74 KDM4E (0.43) HPGDKDM4EEGFRCSF1RALDH1A1
SCHEMBL12755300 0.74 KDM4E (0.40) HPGDKDM4ENQO2ALDH1A1CYP19A1
SCHEMBL12829337 0.74 HPGD (0.43) HPGDKDM4ENQO2ALDH1A1
SCHEMBL29763553 0.74 KDM4E (0.40) HPGDKDM4ENQO2ALDH1A1CYP19A1
SCHEMBL22139831 0.73 EGFR (0.36) EGFRCSF1RALDH1A1
SCHEMBL593723 0.73 KDM4E (0.45) HPGDKDM4ECSF1RNQO2ALDH1A1
SCHEMBL12118481 0.73 EGFR (0.36) EGFRCSF1RALDH1A1
SCHEMBL5779840 0.72 IDO1 (0.49) EGFRCSF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4288424-A1 NOVEL HETEROARYL-SUBSTITUTED IMIDAZOLE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2023-12-13 EP disclosed
WO-2022167631-A1 NOVEL HETEROARYL-SUBSTITUTED IMIDAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2022-08-11 WO disclosed