SCHEMBL29779407

SCHEMBL29779407

O=C1NCC[C@H]1Oc1ccc(Br)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DDB1 Q16531 8/20 0.41
CRBN Q96SW2 8/20 0.41
FPR2 P25090 1/20 0.36
SCN9A Q15858 1/20 0.36
PSEN1 P49768 2/20 0.35
PSEN2 P49810 2/20 0.35
APH1B Q8WW43 2/20 0.35
NCSTN Q92542 2/20 0.35
APH1A Q96BI3 2/20 0.35
PSENEN Q9NZ42 2/20 0.35
ROCK2 O75116 1/20 0.35
PARP10 Q53GL7 2/20 0.33
PARP11 Q9NR21 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
PARP1 P09874 1/20 0.33
HTR2C P28335 1/20 0.33
HTR2B P41595 1/20 0.33
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19297511 1.00 DDB1 (0.41) DDB1CRBNFPR2SCN9APSEN1
SCHEMBL31748160 0.89 PSEN1 (0.42) DDB1CRBNFPR2PSEN1PSEN2
SCHEMBL15632987 0.83 DDB1 (0.41) DDB1CRBNFPR2SCN9A
SCHEMBL4789557 0.83 SLC6A4 (0.44) DDB1CRBNFPR2PSEN1PSEN2
SCHEMBL15632988 0.83 DDB1 (0.41) DDB1CRBNFPR2SCN9A
SCHEMBL20613502 0.83 DDB1 (0.41) DDB1CRBNFPR2SCN9A
SCHEMBL16148496 0.82 DDB1 (0.60) DDB1CRBNROCK2
SCHEMBL16465787 0.80 DDB1 (0.54) DDB1CRBNMAOAMAOB
SCHEMBL15633784 0.80 DDB1 (0.54) DDB1CRBNMAOAMAOB
SCHEMBL15633358 0.80 MCHR1 (0.40) DDB1CRBN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114716370-A Pyridine-containing polycyclic derivative inhibitor, and preparation method and application thereof 上海翰森生物医药科技有限公司 2022-07-08 CN disclosed