SCHEMBL29784145

SCHEMBL29784145

COc1cccc(-c2nc3ccccc3c(=O)[nH]2)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GUSB P08236 4/20 0.73
NPC1 O15118 2/20 0.73
RAB9A P51151 2/20 0.73
TNKS O95271 2/20 0.73
PARP1 P09874 2/20 0.73
TNKS2 Q9H2K2 2/20 0.73
CASP3 P42574 1/20 0.73
SENP7 Q9BQF6 1/20 0.73
SENP6 Q9GZR1 1/20 0.73
CYP1A1 P04798 2/20 0.64
CYP1B1 Q16678 2/20 0.64
CYP1A2 P05177 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL874228 1.00 GUSB (0.73) GUSBNPC1RAB9ATNKSPARP1
SCHEMBL28645325 0.89 GUSB (0.77) GUSBNPC1RAB9ATNKSPARP1
SCHEMBL27694110 0.86 NPC1 (0.61) GUSBNPC1RAB9ATNKSPARP1
SCHEMBL8620410 0.85 TNKS (0.83) GUSBNPC1RAB9ATNKSPARP1
SCHEMBL13011773 0.85 GUSB (0.75) GUSBNPC1RAB9ATNKSPARP1
SCHEMBL17786622 0.85 NPC1 (0.59) GUSBNPC1RAB9ATNKSPARP1
SCHEMBL259622 0.85 KDM4C (0.55) GUSBNPC1RAB9ATNKSPARP1
SCHEMBL27694097 0.85 TNKS (0.58) GUSBNPC1RAB9ATNKSPARP1
SCHEMBL259479 0.85 ALDH1A1 (0.64) GUSBNPC1RAB9ATNKSPARP1
SCHEMBL259476 0.85 KDM4C (0.66) GUSBNPC1RAB9ATNKSPARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118359548-A Preparation method of benzodiazepine compound 重庆医科大学 2024-07-19 CN disclosed
CN-113563272-B Preparation method of 2-phenylquinazolinone compound 三峡大学 2023-03-10 CN disclosed
CN-109879820-B Synthetic method of quinazolinone heterocyclic compound 扬州大学 2022-07-19 CN disclosed