SCHEMBL29790141

SCHEMBL29790141

Cc1cn2c(n1)c(C(N)=O)cc1ccccc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 1/20 0.41
PARP1 P09874 4/20 0.40
TGFBR1 P36897 1/20 0.39
IRAK4 Q9NWZ3 1/20 0.38
AKT1 P31749 1/20 0.38
AKT2 P31751 1/20 0.38
RCE1 Q9Y256 1/20 0.38
ADORA2A P29274 2/20 0.37
ADORA3 P0DMS8 1/20 0.37
ADORA1 P30542 1/20 0.37
SLC9A1 P19634 1/20 0.37
NPC1 O15118 2/20 0.36
MAPT P10636 2/20 0.36
KDM4E B2RXH2 2/20 0.36
GAA P10253 2/20 0.36
MEN1 O00255 1/20 0.36
PABPC1 P11940 1/20 0.36
KMT2A Q03164 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
RAB9A P51151 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29790096 0.81 IKBKB (0.38) IKBKBPARP1TGFBR1IRAK4AKT1
SCHEMBL22902568 0.80 PARP1 (0.41) IKBKBPARP1AKT1AKT2RCE1
SCHEMBL22902800 0.77 ADORA2A (0.45) PARP1IRAK4ADORA2AADORA1NPC1
SCHEMBL29789954 0.75 IKBKB (0.42) IKBKBPARP1IRAK4NPC1MAPT
SCHEMBL19576015 0.74 NNMT (0.39) IKBKBPARP1RCE1ADORA2AADORA3
SCHEMBL22902610 0.72 POLB (0.44) PARP1AKT1AKT2ADORA2AADORA3
SCHEMBL29522831 0.72 POLB (0.44) PARP1AKT1AKT2ADORA2AADORA3
SCHEMBL22902579 0.72 JAK2 (0.36) PARP1RCE1ADORA2AADORA3ADORA1
SCHEMBL4497379 0.70 MEN1 (0.54) IKBKBMAPTKDM4EGAAMEN1
SCHEMBL29790129 0.70 IKBKB (0.42) IKBKBPARP1IRAK4SLC9A1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3999508-A1 TRICYCLIC HETEROARYL COMPOUNDS USEFUL AS IRAK4 INHIBITORS Bristol-Myers Squibb Company (US) 2022-05-25 EP disclosed