SCHEMBL29790484

SCHEMBL29790484

CC(=CC(N)=O)c1nn(COCC[Si](C)(C)C)c2ccc(Br)cc12

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.39
DGAT1 O75907 2/20 0.36
ELANE P08246 8/20 0.35
PDGFRA P16234 1/20 0.34
CDK5 Q00535 1/20 0.34
TYRO3 Q06418 1/20 0.34
IDO1 P14902 2/20 0.32
CFD P00746 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29788710 0.87 ELANE (0.41) NPC1DGAT1ELANETYRO3
SCHEMBL23068015 0.87 ELANE (0.41) NPC1DGAT1ELANETYRO3
SCHEMBL25117904 0.87 ELANE (0.41) NPC1DGAT1ELANETYRO3
SCHEMBL23068016 0.87 ELANE (0.41) NPC1DGAT1ELANETYRO3
SCHEMBL3355071 0.87 NPC1 (0.45) NPC1DGAT1ELANEPDGFRACDK5
SCHEMBL28945073 0.87 DGAT1 (0.40) NPC1DGAT1ELANEPDGFRACDK5
SCHEMBL23068023 0.86 DGAT1 (0.40) NPC1DGAT1ELANEPDGFRACDK5
SCHEMBL492060 0.84 ELANE (0.41) NPC1DGAT1ELANEPDGFRACDK5
SCHEMBL16532624 0.82 ELANE (0.52) NPC1DGAT1ELANEIDO1
SCHEMBL30379746 0.82 ELANE (0.52) NPC1DGAT1ELANEIDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114786673-A CDK inhibitors and their use as medicaments 普莱鲁德疗法有限公司 2022-07-22 CN disclosed