SCHEMBL2979102

SCHEMBL2979102

Cc1ccc(C(=O)Nc2cccc(N3CCOCC3)c2)cc1NC(=O)c1cccc(Cl)c1C

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.56
MAPK14 Q16539 14/20 0.55
SMO Q99835 1/20 0.53
CSF1R P07333 2/20 0.52
NPC1 O15118 1/20 0.52
MAPT P10636 1/20 0.52
NFKB1 P19838 1/20 0.52
NFKB2 Q00653 1/20 0.52
RELA Q04206 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
SETD2 Q9BYW2 1/20 0.51
LCK P06239 1/20 0.51
KDR P35968 1/20 0.51
MAP2K1 Q02750 1/20 0.51
HCK P08631 1/20 0.51
NR2C2 P49116 1/20 0.51
BTK Q06187 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27528929 0.87 MAPK14 (0.59) MAPK14SMOCSF1RSETD2LCK
SCHEMBL2970434 0.84 MAPK14 (0.64) MAPK14SMOCSF1RSETD2LCK
SCHEMBL2975514 0.84 MAPT (0.64) MAPK14SMOCSF1RMAPTSMN1; SMN2
SCHEMBL2979099 0.83 MAPK14 (0.65) RAB9AMAPK14SMOCSF1RSETD2
SCHEMBL6978621 0.82 MAPK14 (0.66) MAPK14
SCHEMBL6782804 0.81 MAPK14 (0.73) RAB9AMAPK14SMOCSF1RNPC1
SCHEMBL14078239 0.81 MAPK14 (0.65) RAB9AMAPK14CSF1RNPC1MAPT
SCHEMBL2972180 0.81 MAPK14 (0.55) MAPK14SMOCSF1RSETD2LCK
SCHEMBL3527294 0.80 MAPK14 (0.62) RAB9AMAPK14SMOCSF1RNPC1
SCHEMBL2969829 0.80 MAPK14 (0.54) MAPK14SMOCSF1RSETD2LCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7772432-B2 Amidobenzamide derivatives which are useful as cytokine inhibitors ASTRAZENECA AB (SE) 2010-08-10 US disclosed
US-20050038081-A1 Amidobenzamide derivatives which are useful as cytokine inhibitors ASTRAZENECA 2005-02-17 US disclosed
US-6821965-B1 IMPORTANT IN DISEASE OR MEDICAL CONDITIONS SUCH AS INFLAMMATION AND IMMUNOREGULATION ASTERZENECA AB (SE) 2004-11-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050038081-A1 Amidobenzamide derivatives which are useful as cytokine inhibitors IL6, IL6ST, IL2 RAB9A 1437/4885MAPK14 1775/4885SMO 4706/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.