SCHEMBL29796402

SCHEMBL29796402

O=CCn1ncc2ccccc21

nearest known ligand 0.56

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
RECQL P46063 2/20 0.56
KMO O15229 1/20 0.54
CYP1A2 P05177 1/20 0.51
DAO P14920 1/20 0.46
ADRA2A P08913 1/20 0.44
POLB P06746 4/20 0.43
NPC1 O15118 4/20 0.42
RAB9A P51151 4/20 0.42
TSHR P16473 3/20 0.42
HSD17B10 Q99714 2/20 0.42
L3MBTL1 Q9Y468 2/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
NPSR1 Q6W5P4 1/20 0.41
P2RX7 Q99572 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3781001 0.82 KMO (0.59) RECQLKMOCYP1A2DAOADRA2A
SCHEMBL29955181 0.82 KMO (0.59) RECQLKMOCYP1A2DAOADRA2A
SCHEMBL3625688 0.81 RECQL (0.56) RECQLKMOCYP1A2DAOADRA2A
SCHEMBL29328565 0.80 KMO (0.56) RECQLKMOCYP1A2DAOADRA2A
SCHEMBL3632921 0.79 FGFR1 (0.42) RECQLKMOCYP1A2
SCHEMBL29411862 0.79 FGFR1 (0.42) RECQLKMOCYP1A2
SCHEMBL3623147 0.79 RECQL (0.53) RECQLKMOCYP1A2DAOADRA2A
SCHEMBL3621969 0.79 RECQL (0.53) RECQLKMOCYP1A2DAOADRA2A
SCHEMBL9934408 0.79 RECQL (0.61) RECQLKMOCYP1A2DAOADRA2A
SCHEMBL323712 0.77 RECQL (0.51) RECQLKMOCYP1A2DAOADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022210479-A1 USE OF AZEPANE DERIVATIVE FOR TREATMENT, AMELIORATION OR PREVENTION OF κ-OPIOID RECEPTOR-RELATED DISEASES 日本ケミファ株式会社 2022-10-06 WO disclosed
CN-114761082-A Azepane derivatives 日本化学药品株式会社 2022-07-15 CN disclosed