SCHEMBL29797178

SCHEMBL29797178

COc1ccc(C(CC(=O)OC(C)(C)C)c2nc(CCCc3ccc4c(n3)NCCC4)co2)cc1F

nearest known ligand 0.61

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ITGAV P06756 19/20 0.61
ITGB3 P05106 17/20 0.61
ITGB6 P18564 11/20 0.61
ITGA2B P08514 6/20 0.61
ITGB5 P18084 5/20 0.51
ITGB8 P26012 5/20 0.51
CXCR4 P61073 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20140591 1.00 ITGAV (0.61) ITGAVITGB3ITGB6ITGA2BITGB5
SCHEMBL20139714 0.93 ITGAV (0.65) ITGAVITGB3ITGB6ITGA2BITGB5
SCHEMBL20139938 0.93 ITGAV (0.65) ITGAVITGB3ITGB6ITGA2BITGB5
SCHEMBL20140538 0.93 ITGAV (0.65) ITGAVITGB3ITGB6ITGA2BITGB5
SCHEMBL20139608 0.83 ITGB3 (0.40) ITGAVITGB3ITGB6ITGA2BITGB5
SCHEMBL29797182 0.83 ITGB3 (0.40) ITGAVITGB3ITGB6ITGA2BITGB5
SCHEMBL20140195 0.83 ITGAV (0.54) ITGAVITGB3ITGB6ITGA2BITGB5
SCHEMBL29797306 0.83 ITGAV (0.54) ITGAVITGB3ITGB6ITGA2BITGB5
SCHEMBL20142767 0.81 ITGB3 (0.40) ITGAVITGB3ITGB6ITGA2B
SCHEMBL29797239 0.81 ITGB3 (0.40) ITGAVITGB3ITGB6ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110167935-B 3-substituted propionic acids as alpha V integrin inhibitors 百时美施贵宝公司 2022-05-27 CN disclosed