SCHEMBL29797429

SCHEMBL29797429

CCOC(=O)CC(c1ccc(OC)c(F)c1)c1nc(Br)cs1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CTSA P10619 12/20 0.40
PRKCZ Q05513 1/20 0.40
RAB9A P51151 2/20 0.38
ITGB3 P05106 1/20 0.38
ITGAV P06756 1/20 0.38
ITGA2B P08514 1/20 0.38
ITGB6 P18564 1/20 0.38
NPC1 O15118 1/20 0.38
FFAR1 O14842 1/20 0.37
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
MAPK1 P28482 1/20 0.36
HTT P42858 1/20 0.36
ABCB1 P08183 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20139522 1.00 CTSA (0.40) CTSAPRKCZRAB9AITGB3ITGAV
SCHEMBL20140402 0.81 CTSA (0.41) CTSAITGB3ITGAVITGB6FFAR1
SCHEMBL29797198 0.79 FGFR2 (0.38) CTSAPRKCZRAB9AITGB3ITGAV
SCHEMBL20139722 0.79 FGFR2 (0.38) CTSAPRKCZRAB9AITGB3ITGAV
SCHEMBL29797153 0.78 CTSA (0.41) CTSARAB9ANPC1FFAR1LMNA
SCHEMBL20139502 0.78 CTSA (0.41) CTSARAB9ANPC1FFAR1LMNA
SCHEMBL20380272 0.75 FFAR1 (0.44) PRKCZRAB9AFFAR1ALDH1A1LMNA
SCHEMBL29797272 0.75 ITGB3 (0.47) CTSAPRKCZRAB9AITGB3ITGAV
SCHEMBL20139498 0.75 ITGB3 (0.47) CTSAPRKCZRAB9AITGB3ITGAV
SCHEMBL20139800 0.74 ITGB3 (0.44) CTSAPRKCZRAB9AITGB3ITGAV

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110167935-B 3-substituted propionic acids as alpha V integrin inhibitors 百时美施贵宝公司 2022-05-27 CN disclosed