SCHEMBL298053

SCHEMBL298053

FC(F)(F)c1nnc(-c2cccs2)s1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 13/20 0.56
ALDH1A1 P00352 10/20 0.56
HSD17B10 Q99714 6/20 0.56
EPHX2 P34913 1/20 0.56
RAB9A P51151 9/20 0.47
SMN1; SMN2 Q16637 6/20 0.47
KMT2A Q03164 3/20 0.47
RECQL P46063 1/20 0.47
HPGD P15428 7/20 0.43
NPC1 O15118 6/20 0.43
PKM P14618 1/20 0.43
GAA P10253 1/20 0.42
LMNA P02545 1/20 0.42
HTT P42858 1/20 0.42
NLRP1 Q9C000 1/20 0.42
L3MBTL1 Q9Y468 2/20 0.41
MEN1 O00255 1/20 0.41
MAPT P10636 1/20 0.41
CASP3 P42574 1/20 0.41
SENP8 Q96LD8 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL298901 0.90 KDM4E (0.46) KDM4EALDH1A1HSD17B10EPHX2RAB9A
SCHEMBL11991177 0.80 KDM4E (0.73) KDM4EALDH1A1HSD17B10EPHX2RAB9A
SCHEMBL971554 0.72 KDM4E (0.61) KDM4EALDH1A1HSD17B10EPHX2RAB9A
SCHEMBL6374937 0.72 KDM4E (1.00) KDM4EALDH1A1HSD17B10EPHX2RAB9A
SCHEMBL11701666 0.72 KDM4E (0.61) KDM4EALDH1A1HSD17B10EPHX2RAB9A
SCHEMBL28723226 0.70 KDM4E (0.59) KDM4EALDH1A1HSD17B10EPHX2RAB9A
SCHEMBL28719243 0.70 KDM4E (0.59) KDM4EALDH1A1HSD17B10EPHX2RAB9A
SCHEMBL27914246 0.70 KDM4E (0.96) KDM4EALDH1A1HSD17B10EPHX2RAB9A
SCHEMBL10495079 0.68 KDM4E (0.51) KDM4EALDH1A1HSD17B10EPHX2RAB9A
SCHEMBL11631549 0.67 KDM4E (0.54) KDM4EALDH1A1HSD17B10EPHX2RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103288776-B A synthesis method for 2 - sulfinyl -5 - (trifluoromethyl) - 1,3,4 - thiadiazole compounds ZHEJIANG ZHUJI UNITED CHEMICALS CO LTD 2015-05-13 CN disclosed
CN-103288776-A A synthesis method for 2 - sulfinyl -5 - (trifluoromethyl) - 1,3,4 - thiadiazole compounds ZHEJIANG ZHUJI UNITED CHEMICALS CO LTD 2013-09-11 CN disclosed
EP-2427447-A2 SMALL MOLECULE INHIBITORS OF INFLUENZA A AND B VIRUS AND RESPIRATORY SYNCYTIAL VIRUS REPLICATION Pike Pharma GmbH (CH) 2012-03-14 EP disclosed
WO-2010128163-A2 SMALL MOLECULE INHIBITORS OF INFLUENZA A AND B VIRUS AND RESPIRATORY SYNCYTIAL VIRUS REPLICATION PIKE PHARMA GMBH (CH) 2010-11-11 WO disclosed