SCHEMBL298901

SCHEMBL298901

FC(F)(F)c1nnc(-c2ccc(-c3cccs3)s2)s1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.46
ALDH1A1 P00352 6/20 0.46
HSD17B10 Q99714 3/20 0.46
EPHX2 P34913 1/20 0.46
DPP4 P27487 4/20 0.41
RAB9A P51151 5/20 0.40
SMN1; SMN2 Q16637 5/20 0.40
KMT2A Q03164 2/20 0.40
RECQL P46063 1/20 0.40
LTA4H P09960 1/20 0.39
NPC1 O15118 3/20 0.37
HPGD P15428 2/20 0.37
HDAC1 Q13547 2/20 0.37
PKM P14618 1/20 0.37
HDAC3 O15379 1/20 0.37
HDAC4 P56524 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
GAA P10253 3/20 0.37
LMNA P02545 2/20 0.37
L3MBTL1 Q9Y468 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL298053 0.90 KDM4E (0.56) KDM4EALDH1A1HSD17B10EPHX2RAB9A
SCHEMBL298601 0.76 KDM4E (0.50) KDM4EALDH1A1HSD17B10EPHX2DPP4
SCHEMBL299482 0.74 APP (0.38) ALDH1A1
SCHEMBL2742433 0.73 DPP4 (0.65) KDM4EALDH1A1HSD17B10EPHX2DPP4
Alpha-Terthienyl SCHEMBL147274 0.73 DPP4 (0.65) KDM4EALDH1A1HSD17B10EPHX2DPP4
SCHEMBL23611278 0.73 DPP4 (0.65) KDM4EALDH1A1HSD17B10EPHX2DPP4
SCHEMBL14703073 0.73 DPP4 (0.65) KDM4EALDH1A1HSD17B10EPHX2DPP4
SCHEMBL499333 0.73 DPP4 (0.65) KDM4EALDH1A1HSD17B10EPHX2DPP4
SCHEMBL13707354 0.73 DPP4 (0.65) KDM4EALDH1A1HSD17B10EPHX2DPP4
SCHEMBL1105086 0.73 DPP4 (0.65) KDM4EALDH1A1HSD17B10EPHX2DPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427447-A2 SMALL MOLECULE INHIBITORS OF INFLUENZA A AND B VIRUS AND RESPIRATORY SYNCYTIAL VIRUS REPLICATION Pike Pharma GmbH (CH) 2012-03-14 EP disclosed
WO-2010128163-A2 SMALL MOLECULE INHIBITORS OF INFLUENZA A AND B VIRUS AND RESPIRATORY SYNCYTIAL VIRUS REPLICATION PIKE PHARMA GMBH (CH) 2010-11-11 WO disclosed