SCHEMBL29807993

SCHEMBL29807993

Cc1csc2nccc(O)c12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MRGPRX1 Q96LB2 1/20 0.38
HTT P42858 2/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
LMNA P02545 2/20 0.36
POLB P06746 1/20 0.36
GAA P10253 1/20 0.36
PKM P14618 1/20 0.36
PIP4K2C Q8TBX8 1/20 0.35
LIMK1 P53667 1/20 0.35
ESR1 P03372 1/20 0.35
IRAK4 Q9NWZ3 1/20 0.33
PDK1 Q15118 3/20 0.32
CTDSP1 Q9GZU7 1/20 0.32
ALOX12 P18054 1/20 0.31
HSP90AA1 P07900 1/20 0.31
CCR6 P51684 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
SLC6A2 P23975 1/20 0.31
ELANE P08246 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1904104 1.00 MRGPRX1 (0.38) MRGPRX1HTTRAB9ASMN1; SMN2LMNA
SCHEMBL13460085 0.82 HTT (0.42) MRGPRX1HTTRAB9ASMN1; SMN2LMNA
SCHEMBL28381075 0.77 HTT (0.40) MRGPRX1HTTRAB9ASMN1; SMN2LMNA
SCHEMBL1899302 0.77 MRGPRX1 (0.38) MRGPRX1HTTRAB9ASMN1; SMN2LMNA
SCHEMBL27023187 0.74 RAB9A (0.38) MRGPRX1HTTRAB9ASMN1; SMN2LMNA
SCHEMBL25636165 0.74 MRGPRX1 (0.36) MRGPRX1HTTRAB9ASMN1; SMN2LMNA
SCHEMBL1604974 0.72 MRGPRX1 (0.46) MRGPRX1HTTRAB9ASMN1; SMN2LMNA
SCHEMBL25030030 0.71 HTR2A (0.44)
SCHEMBL25028223 0.71 HTR2A (0.41) HTTRAB9ASMN1; SMN2LMNA
SCHEMBL1330351 0.71 PDPK1 (0.44) HTTRAB9APKMSLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4277892-A1 SPIROCYCLOHEXANE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR USES AS ANTI-APOPTOTIC INHIBITORS Les Laboratoires Servier (FR) 2023-11-22 EP disclosed
WO-2022152705-A1 SPIROCYCLOHEXANE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR USES AS ANTI-APOPTOTIC INHIBITORS LES LABORATOIRES SERVIER (FR) 2022-07-21 WO disclosed