SCHEMBL29809100

SCHEMBL29809100

O=[N+]([O-])c1c(Cl)nc2ccccc2c1NCc1ccc(CN2CCCC2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.53
PKM P14618 1/20 0.45
ACP1 P24666 1/20 0.45
ACHE P22303 4/20 0.45
ALDH1A1 P00352 3/20 0.44
HPGD P15428 2/20 0.44
BCHE P06276 2/20 0.44
BACE1 P56817 2/20 0.44
KDM4E B2RXH2 1/20 0.43
MAPT P10636 1/20 0.43
MAPK1 P28482 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
LMNA P02545 1/20 0.43
KMT2A Q03164 2/20 0.43
POLB P06746 1/20 0.43
RAD52 P43351 1/20 0.43
MEN1 O00255 1/20 0.41
HRH3 Q9Y5N1 1/20 0.41
CCR2 P41597 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24732868 1.00 EGFR (0.53) EGFRPKMACP1ACHEALDH1A1
SCHEMBL24732595 0.92 EGFR (0.45) EGFRACP1ACHEALDH1A1HPGD
SCHEMBL29809575 0.92 EGFR (0.45) EGFRACP1ACHEALDH1A1HPGD
SCHEMBL29809351 0.91 EGFR (0.44) EGFRACP1ACHEALDH1A1HPGD
SCHEMBL24732862 0.91 EGFR (0.44) EGFRACP1ACHEALDH1A1HPGD
SCHEMBL24733000 0.90 EGFR (0.43) EGFRALDH1A1HPGDKDM4EMAPT
SCHEMBL29809025 0.90 EGFR (0.43) EGFRALDH1A1HPGDKDM4EMAPT
SCHEMBL24733032 0.90 EGFR (0.45) EGFRPKMACP1ACHEALDH1A1
SCHEMBL24732827 0.90 EGFR (0.45) EGFRPKMACP1ACHEALDH1A1
SCHEMBL29809050 0.90 EGFR (0.45) EGFRPKMACP1ACHEALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117736210-A Aromatic heterocyclic compound, and preparation method and application thereof 上海翊石医药科技有限公司 2024-03-22 CN disclosed
CN-114805341-B Aromatic heterocyclic compound, and preparation method and application thereof 上海翊石医药科技有限公司 2023-12-08 CN disclosed
CN-114805341-A Aromatic heterocyclic compounds and preparation method and application thereof 上海翊石医药科技有限公司 2022-07-29 CN disclosed