SCHEMBL29809351

SCHEMBL29809351

O=[N+]([O-])c1c(Cl)nc2ccccc2c1NCc1cccc(CN2CCCCC2)c1

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.44
PDE5A O76074 1/20 0.43
ACP1 P24666 4/20 0.42
ACHE P22303 1/20 0.41
MAP3K7 O43318 1/20 0.41
IRAK1 P51617 1/20 0.41
IRAK4 Q9NWZ3 1/20 0.41
ALDH1A1 P00352 4/20 0.41
MAPT P10636 3/20 0.41
POLB P06746 2/20 0.41
KDM4E B2RXH2 2/20 0.41
MAPK1 P28482 2/20 0.41
HPGD P15428 1/20 0.41
LMNA P02545 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
MAOB P27338 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
NPSR1 Q6W5P4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24732862 1.00 EGFR (0.44) EGFRPDE5AACP1ACHEMAP3K7
SCHEMBL24732595 0.99 EGFR (0.45) EGFRPDE5AACP1ACHEALDH1A1
SCHEMBL29809575 0.99 EGFR (0.45) EGFRPDE5AACP1ACHEALDH1A1
SCHEMBL29809100 0.91 EGFR (0.53) EGFRACP1ACHEALDH1A1MAPT
SCHEMBL24732868 0.91 EGFR (0.53) EGFRACP1ACHEALDH1A1MAPT
SCHEMBL24733021 0.91 LMNA (0.44) EGFRPDE5AACP1ALDH1A1MAPT
SCHEMBL29809290 0.91 EGFR (0.45) EGFRPDE5AACP1ALDH1A1MAPT
SCHEMBL24733480 0.91 EGFR (0.45) EGFRPDE5AACP1ALDH1A1MAPT
SCHEMBL29809120 0.91 LMNA (0.44) EGFRPDE5AACP1ALDH1A1MAPT
SCHEMBL24732670 0.88 CACNB4 (0.45) ACHEALDH1A1MAPTPOLBKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114805341-B Aromatic heterocyclic compound, and preparation method and application thereof 上海翊石医药科技有限公司 2023-12-08 CN disclosed
CN-114805341-A Aromatic heterocyclic compounds and preparation method and application thereof 上海翊石医药科技有限公司 2022-07-29 CN disclosed