SCHEMBL29809266

SCHEMBL29809266

Nc1c(Cl)nc2cccc(Cc3cccc(Cn4cccn4)c3)c2c1N

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.41
MEN1 O00255 1/20 0.38
TSHR P16473 1/20 0.38
KMT2A Q03164 1/20 0.38
GAA P10253 1/20 0.38
MAPT P10636 1/20 0.38
PRKACA P17612 1/20 0.37
PRKACG P22612 1/20 0.37
PRKACB P22694 1/20 0.37
KLKB1 P03952 1/20 0.37
KLK1 P06870 1/20 0.37
GLS O94925 3/20 0.36
NOS3 P29474 1/20 0.36
NOS1 P29475 1/20 0.36
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA9 Q16790 1/20 0.36
HDAC1 Q13547 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28802745 1.00 HTT (0.41) HTTMEN1TSHRKMT2AGAA
SCHEMBL213846 0.78 DHFR (0.46) HTTMEN1KMT2AMPOCYP3A4
SCHEMBL29978287 0.74 APP (0.43) HTTMEN1TSHRKMT2APRKACA
SCHEMBL24732797 0.74 APP (0.43) HTTMEN1TSHRKMT2APRKACA
SCHEMBL28802703 0.73 TLR8 (0.34) NOS3NOS1TLR8
SCHEMBL29809381 0.73 TLR8 (0.34) NOS3NOS1TLR8
SCHEMBL15081591 0.73 HTT (0.61) HTTMEN1TSHRKMT2AGAA
SCHEMBL14256403 0.72 HTT (0.68) HTTMEN1TSHRKMT2AGAA
SCHEMBL16347168 0.68 HTT (0.59) HTTMEN1TSHRKMT2AGAA
SCHEMBL1851019 0.68 HTT (0.59) HTTMEN1TSHRKMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114805341-B Aromatic heterocyclic compound, and preparation method and application thereof 上海翊石医药科技有限公司 2023-12-08 CN disclosed
CN-114805341-A Aromatic heterocyclic compounds and preparation method and application thereof 上海翊石医药科技有限公司 2022-07-29 CN disclosed