SCHEMBL29834784

SCHEMBL29834784

Nc1ccc(Oc2ccnc(N3CCCC3)c2)cc1F

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 1/20 0.39
CCR6 P51684 1/20 0.39
CNR2 P34972 2/20 0.39
NFKB1 P19838 2/20 0.38
NR2C2 P49116 2/20 0.38
NFKB2 Q00653 2/20 0.38
RELA Q04206 2/20 0.38
TAB1 Q15750 2/20 0.38
CCNC P24863 1/20 0.37
CDK8 P49336 1/20 0.37
NMT1 P30419 1/20 0.36
LRRK2 Q5S007 2/20 0.36
MAPK13 O15264 1/20 0.35
NR4A1 P22736 1/20 0.35
CXCR4 P61073 1/20 0.35
ELOVL1 Q9BW60 1/20 0.34
TNK2 Q07912 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29834720 0.99 HRH4 (0.41) HRH4CCR6CNR2NFKB1NR2C2
SCHEMBL24037401 0.88 MAPK13 (0.47) CNR2LRRK2MAPK13ELOVL1
SCHEMBL27096991 0.83 LRRK2 (0.39) LRRK2
SCHEMBL27096964 0.82 OPRD1 (0.35) CCR6NMT1LRRK2
SCHEMBL27096891 0.81 LRRK2 (0.43) CCR6LRRK2NR4A1
SCHEMBL11958457 0.81 NR4A1 (0.37) NR4A1
SCHEMBL29834771 0.80 LRRK2 (0.43) LRRK2
SCHEMBL29834781 0.80 TYK2 (0.36) MAPK13
SCHEMBL29834705 0.80 MAP4K4 (0.43) CCNCCDK8LRRK2
SCHEMBL11958458 0.80 NR4A1 (0.36) NR4A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022170043-A1 QUINAZOLINE DERIVED COMPOUNDS AS EGFR INHIBITORS AND THEIR USES THEREOF ACCUTAR BIOTECHNOLOGY, INC. (US) 2022-08-11 WO disclosed