SCHEMBL29849809

SCHEMBL29849809

NC(=O)c1ccncc1-c1ccc2c(c1)CC(=O)N2

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 2/20 0.59
PDE3A Q14432 2/20 0.59
CYP11B2 P19099 4/20 0.56
CYP11B1 P15538 3/20 0.56
CYP1A2 P05177 2/20 0.56
CRBN Q96SW2 1/20 0.49
GRIA1 P42261 6/20 0.48
CACNG8 Q8WXS5 2/20 0.48
AOC2 O75106 1/20 0.44
SYK P43405 1/20 0.44
CYP2C9 P11712 2/20 0.43
TBXAS1 P24557 1/20 0.43
PGR P06401 1/20 0.43
TDP2 O95551 1/20 0.43
JAK3 P52333 1/20 0.42
IRAK4 Q9NWZ3 1/20 0.42
BMPR1B O00238 1/20 0.42
BMPR1A P36894 1/20 0.42
TGFBR1 P36897 1/20 0.42
ACVRL1 P37023 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7076084 0.82 GRIA1 (0.63) PDE3BPDE3ACYP11B2CYP11B1CYP1A2
SCHEMBL29849879 0.80 GRIA1 (0.67) PDE3BPDE3ACYP11B2CYP11B1CYP1A2
SCHEMBL26463255 0.80 GRIA1 (0.67) PDE3BPDE3ACYP11B2CYP11B1CYP1A2
SCHEMBL29850035 0.77 PDE3B (0.60) PDE3BPDE3ACYP11B2CYP11B1CYP1A2
SCHEMBL23143482 0.75 PDE3B (1.00) PDE3BPDE3ACYP11B2CYP11B1CYP1A2
SCHEMBL31139508 0.72 GRIA1 (0.50) PDE3BPDE3ACYP11B2CYP11B1CYP1A2
SCHEMBL29899595 0.72 CYP11B1 (1.00) PDE3BPDE3ACYP11B2CYP11B1CYP1A2
SCHEMBL29849827 0.72 CYP11B1 (1.00) PDE3BPDE3ACYP11B2CYP11B1CYP1A2
SCHEMBL748904 0.72 CYP11B1 (1.00) PDE3BPDE3ACYP11B2CYP11B1CYP1A2
SCHEMBL29849907 0.72 CYP11B1 (1.00) PDE3BPDE3ACYP11B2CYP11B1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4034526-A1 THERAPEUTIC COMPOUNDS AND METHODS OF USE THEREOF Agency for Science, Technology and Research (A*STAR) (SG) 2022-08-03 EP disclosed