SCHEMBL29856174

SCHEMBL29856174

C#Cc1cc(C(=O)Nc2ccc(CN3CCN(CCO)CC3)c(F)c2)ccc1C

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIT P10721 6/20 0.68
ABL1 P00519 12/20 0.55
SRC P12931 2/20 0.55
FGFR1 P11362 2/20 0.55
KDR P35968 2/20 0.55
JAK2 O60674 1/20 0.55
EGFR P00533 1/20 0.55
RET P07949 1/20 0.55
PDGFRB P09619 1/20 0.55
BRAF P15056 1/20 0.55
PDGFRA P16234 1/20 0.55
FLT1 P17948 1/20 0.55
FGFR2 P21802 1/20 0.55
FGFR4 P22455 1/20 0.55
FGFR3 P22607 1/20 0.55
JAK1 P23458 1/20 0.55
CCNE1 P24864 1/20 0.55
CDK2 P24941 1/20 0.55
EPHA2 P29317 1/20 0.55
EPHA3 P29320 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22288302 1.00 KIT (0.68) KITABL1SRCFGFR1KDR
SCHEMBL29856255 0.93 KIT (0.78) KITABL1FGFR1KDRBRAF
SCHEMBL16755338 0.93 KIT (0.78) KITABL1FGFR1KDRBRAF
SCHEMBL16755299 0.88 KIT (0.87) KITABL1SRCFGFR1KDR
SCHEMBL28439198 0.84 KIT (0.79) KITABL1FGFR1KDRBRAF
SCHEMBL29856195 0.84 KIT (0.79) KITABL1FGFR1KDRBRAF
SCHEMBL13813508 0.82 KIT (0.77) KITABL1FGFR1KDRBRAF
SCHEMBL22300440 0.81 KIT (0.61) KITABL1FGFR1KDRRET
SCHEMBL22300432 0.81 KIT (0.61) KITABL1FGFR1KDRRET
SCHEMBL28441871 0.81 KIT (0.61) KITABL1FGFR1KDRRET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111484482-B Alkynyl pyrimidine or alkynyl pyridine compound, and composition and application thereof 北京赛特明强医药科技有限公司 2022-06-21 CN disclosed