SCHEMBL29857044

SCHEMBL29857044

O=C(Nc1cccnc1)c1cc(-c2cnn(CCN3CCOCC3)c2)ccc1OCc1ccc(F)cc1

nearest known ligand 0.76

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 16/20 0.76
SRPK3 Q9UPE1 1/20 0.57
IKBKE Q14164 1/20 0.54
TBK1 Q9UHD2 1/20 0.54
SGMS2 Q8NHU3 2/20 0.49
GSK3B P49841 1/20 0.47
DYRK1A Q13627 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6918063 1.00 LRRK2 (0.76) LRRK2SRPK3IKBKETBK1SGMS2
SCHEMBL25951821 0.93 LRRK2 (0.65) LRRK2SRPK3IKBKETBK1
SCHEMBL1646947 0.90 LRRK2 (0.61) LRRK2IKBKETBK1GSK3BDYRK1A
SCHEMBL6916617 0.88 LRRK2 (0.83) LRRK2SRPK3SGMS2
SCHEMBL28347793 0.88 LRRK2 (0.57) LRRK2SRPK3IKBKETBK1
SCHEMBL1648915 0.87 LRRK2 (0.82) LRRK2SRPK3IKBKETBK1SGMS2
SCHEMBL1647667 0.87 LRRK2 (1.00) LRRK2SRPK3SGMS2
SCHEMBL10322929 0.85 LRRK2 (0.63) LRRK2SRPK3SGMS2
SCHEMBL6917908 0.84 LRRK2 (0.67) LRRK2SRPK3SGMS2
SCHEMBL1646768 0.84 LRRK2 (0.51) LRRK2IKBKETBK1GSK3BDYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110678182-B Pharmaceutical composition containing a compound capable of penetrating the blood-brain barrier as an active ingredient for preventing or treating brain cancer 大邱庆北尖端医疗产业振兴财团 2022-08-23 CN disclosed