SCHEMBL29860116

SCHEMBL29860116

O=C1Nc2c(ccc(F)c2F)C1=O

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CES1 P23141 9/20 0.50
TGM2 P21980 3/20 0.50
DAO P14920 2/20 0.46
NSD2 O96028 1/20 0.46
BCHE P06276 1/20 0.46
LIG1 P18858 1/20 0.42
DNMT1 P26358 1/20 0.41
CASP3 P42574 1/20 0.39
CASP2 P42575 1/20 0.39
CASP7 P55210 1/20 0.39
CASP6 P55212 1/20 0.39
CASP8 Q14790 1/20 0.39
MAOA P21397 2/20 0.38
MAOB P27338 2/20 0.38
GRM5 P41594 1/20 0.36
ALDH1A1 P00352 1/20 0.35
ALDH2 P05091 1/20 0.35
ALDH3A1 P30838 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3076875 1.00 CES1 (0.50) CES1TGM2DAONSD2BCHE
SCHEMBL3085898 0.80 CES1 (0.62) CES1TGM2DAONSD2BCHE
SCHEMBL29689346 0.80 CES1 (0.62) CES1TGM2DAONSD2BCHE
SCHEMBL2661276 0.80 CES1 (0.47) CES1TGM2DAONSD2BCHE
SCHEMBL14358786 0.80 CES1 (0.67) CES1TGM2DAONSD2BCHE
SCHEMBL29689423 0.80 CES1 (0.67) CES1TGM2DAONSD2BCHE
SCHEMBL2373643 0.80 CES1 (0.47) CES1TGM2DAONSD2BCHE
SCHEMBL3093497 0.80 DAO (0.56) CES1TGM2DAONSD2BCHE
SCHEMBL15228756 0.80 CES1 (0.47) CES1TGM2DAONSD2BCHE
SCHEMBL30441928 0.80 CES1 (0.67) CES1TGM2DAONSD2BCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119330941-A Antitumor compounds as UPR agonists and uses thereof 南京圣和药业股份有限公司 2025-01-21 CN disclosed
EP-4452937-A1 COMPOUNDS Psylo Pty Ltd (AU) 2024-10-30 EP disclosed
CN-118812517-A Antitumor compounds as UPR agonists and uses thereof 南京圣和药业股份有限公司 2024-10-22 CN disclosed
CN-118715204-A Compounds of formula (I) 普赛洛私人有限公司 2024-09-27 CN disclosed
WO-2024175114-A1 BORON CONTAINING COMPOUNDS AND THERAPEUTIC USES THEREOF Shanghai Yuyao Biotech Ltd. (CN) 2024-08-29 WO disclosed
CN-116997550-A N- (benzoyl) -phenylalanine compounds, pharmaceutical compositions containing same and application thereof 杭州普洛药物研究院有限公司 2023-11-03 CN disclosed
WO-2023115166-A1 COMPOUNDS Psylo Pty Ltd (AU) 2023-06-29 WO disclosed
CN-114853659-A N- (benzoyl) -phenylalanine compounds, pharmaceutical compositions containing same, and uses thereof 普洛药业股份有限公司 2022-08-05 CN disclosed