SCHEMBL29862404

SCHEMBL29862404

C[Si](C)(C)CCOCn1c(-c2ccnc3[nH]ccc23)cc(C(N)=O)c1-c1cccc(Cl)c1F

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NUDT1 P36639 2/20 0.42
PRKCI P41743 1/20 0.39
JAK2 O60674 4/20 0.38
JAK1 P23458 4/20 0.38
TYK2 P29597 3/20 0.38
IKBKB O14920 1/20 0.37
CHUK O15111 1/20 0.37
CCNK O75909 1/20 0.36
CDK12 Q9NYV4 1/20 0.36
RHEB Q15382 1/20 0.36
CIT O14578 5/20 0.36
MAPK14 Q16539 1/20 0.35
NPC1 O15118 1/20 0.35
BRAF P15056 2/20 0.34
TNIK Q9UKE5 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27282728 1.00 NUDT1 (0.42) NUDT1PRKCIJAK2JAK1TYK2
SCHEMBL29862246 0.93 RHEB (0.38) NUDT1PRKCIJAK2JAK1TYK2
SCHEMBL27282657 0.93 RHEB (0.38) NUDT1PRKCIJAK2JAK1TYK2
SCHEMBL27282737 0.92 NUDT1 (0.43) NUDT1PRKCIJAK2JAK1TYK2
SCHEMBL27282734 0.92 NUDT1 (0.43) NUDT1PRKCIJAK2JAK1TYK2
SCHEMBL27282755 0.92 NUDT1 (0.43) NUDT1PRKCIJAK2JAK1TYK2
SCHEMBL27282753 0.91 NUDT1 (0.42) NUDT1PRKCIJAK2JAK1TYK2
SCHEMBL27282749 0.91 NUDT1 (0.42) NUDT1PRKCIJAK2JAK1TYK2
SCHEMBL29862299 0.90 NUDT1 (0.42) NUDT1PRKCIJAK2JAK1TYK2
SCHEMBL27282773 0.90 NUDT1 (0.42) NUDT1PRKCIJAK2JAK1TYK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4313971-A1 SUBSTITUTED PYRROLE CARBOXAMIDES, PROCESS FOR THEIR PREPARATION AND THEIR USE AS KINASE INHIBITORS Nerviano Medical Sciences S.r.l. (IT) 2024-02-07 EP disclosed
CN-117157289-A Substituted pyrrolecarboxamides, process for their preparation and their use as kinase inhibitors 内尔维亚诺医疗科学公司 2023-12-01 CN disclosed
WO-2022207404-A1 SUBSTITUTED PYRROLE CARBOXAMIDES, PROCESS FOR THEIR PREPARATION AND THEIR USE AS KINASE INHIBITORS NERVIANO MEDICAL SCIENCES S.R.L. (IT) 2022-10-06 WO disclosed