SCHEMBL29862939

SCHEMBL29862939

O=C(O)Cn1cc(-c2cccc(NC(=O)c3cccc(Cl)c3)c2)nn1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.56
KDM4E B2RXH2 1/20 0.56
ALDH1A1 P00352 1/20 0.56
LMNA P02545 1/20 0.56
MAPT P10636 1/20 0.56
CDC7 O00311 1/20 0.54
DAPK3 O43293 1/20 0.54
PAK4 O96013 1/20 0.54
CDK2 P24941 1/20 0.54
FLT3 P36888 1/20 0.54
CSNK1A1 P48729 1/20 0.54
CLK2 P49760 1/20 0.54
GSK3B P49841 1/20 0.54
CDK7 P50613 1/20 0.54
CDK9 P50750 1/20 0.54
PRKX P51817 1/20 0.54
CDK5 Q00535 1/20 0.54
DYRK1A Q13627 1/20 0.54
MELK Q14680 1/20 0.54
HIPK2 Q9H2X6 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28396447 1.00 KMT2A (0.56) KMT2AKDM4EALDH1A1LMNAMAPT
SCHEMBL22566519 0.89 HDAC3 (0.70) KMT2AKDM4EALDH1A1LMNAMAPT
SCHEMBL29862961 0.88 TP53 (0.53) KMT2AKDM4EALDH1A1LMNAMAPT
SCHEMBL28401956 0.88 TP53 (0.53) KMT2AKDM4EALDH1A1LMNAMAPT
SCHEMBL22566549 0.86 TSHR (0.63) KMT2AALDH1A1LMNAMAPTCDC7
SCHEMBL29862908 0.85 HDAC3 (0.54) KMT2AKDM4EALDH1A1LMNACDC7
SCHEMBL28400450 0.85 HDAC3 (0.54) KMT2AKDM4EALDH1A1LMNACDC7
SCHEMBL28397320 0.84 TP53 (0.52) KMT2AKDM4EALDH1A1LMNAHDAC3
SCHEMBL29863344 0.84 TP53 (0.52) KMT2AKDM4EALDH1A1LMNAHDAC3
SCHEMBL29863155 0.82 KDM4E (0.60) KMT2AKDM4EALDH1A1LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111057015-B 2- (4-phenyl-1H-1, 2, 3-triazole-1-yl) acetic acid and acethydrazide compounds 中国医科大学 2022-09-16 CN claimed
CN-111057015-B 2- (4-phenyl-1H-1, 2, 3-triazole-1-yl) acetic acid and acethydrazide compounds 中国医科大学 2022-09-16 CN disclosed