SCHEMBL29863155

SCHEMBL29863155

COc1ccc(C(=O)Nc2cccc(-c3cn(CC(=O)O)nn3)c2)cc1OC

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.60
SMN1; SMN2 Q16637 1/20 0.60
POLB P06746 4/20 0.58
MAPT P10636 3/20 0.58
TP53 P04637 1/20 0.58
NPC1 O15118 2/20 0.55
RAB9A P51151 2/20 0.55
SRC P12931 2/20 0.54
CDC7 O00311 1/20 0.54
PLK4 O00444 1/20 0.54
CHEK1 O14757 1/20 0.54
AURKA O14965 1/20 0.54
DCLK1 O15075 1/20 0.54
MAPK13 O15264 1/20 0.54
PDPK1 O15530 1/20 0.54
DAPK3 O43293 1/20 0.54
DYRK3 O43781 1/20 0.54
JAK2 O60674 1/20 0.54
ROCK2 O75116 1/20 0.54
PRKD3 O94806 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28403964 1.00 KDM4E (0.60) KDM4ESMN1; SMN2POLBMAPTTP53
SCHEMBL22566549 0.88 TSHR (0.63) SMN1; SMN2POLBMAPTTP53NPC1
SCHEMBL28400450 0.84 HDAC3 (0.54) KDM4ESMN1; SMN2POLBTP53RAB9A
SCHEMBL29862908 0.84 HDAC3 (0.54) KDM4ESMN1; SMN2POLBTP53RAB9A
SCHEMBL28397320 0.83 TP53 (0.52) KDM4ESMN1; SMN2POLBTP53NPC1
SCHEMBL29863344 0.83 TP53 (0.52) KDM4ESMN1; SMN2POLBTP53NPC1
SCHEMBL29862939 0.82 KMT2A (0.56) KDM4EPOLBMAPTNPC1RAB9A
SCHEMBL28401956 0.82 TP53 (0.53) KDM4ESMN1; SMN2MAPTTP53NPC1
SCHEMBL28396447 0.82 KMT2A (0.56) KDM4EPOLBMAPTNPC1RAB9A
SCHEMBL29862961 0.82 TP53 (0.53) KDM4ESMN1; SMN2MAPTTP53NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111057015-B 2- (4-phenyl-1H-1, 2, 3-triazole-1-yl) acetic acid and acethydrazide compounds 中国医科大学 2022-09-16 CN disclosed