SCHEMBL29863036

SCHEMBL29863036

COc1cc(N[C@@H]2CCNC2)c2cccnc2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 5/20 0.46
CHEK1 O14757 4/20 0.46
MAOB P27338 1/20 0.42
HTR6 P50406 1/20 0.42
MKNK1 Q9BUB5 1/20 0.41
MKNK2 Q9HBH9 1/20 0.41
AXL P30530 1/20 0.41
CYP1A2 P05177 3/20 0.41
LMNA P02545 2/20 0.41
CYP3A4 P08684 2/20 0.41
MAPK1 P28482 2/20 0.41
HSD17B10 Q99714 2/20 0.41
ALDH1A1 P00352 1/20 0.41
TP53 P04637 1/20 0.41
ALOX15 P16050 1/20 0.41
TSHR P16473 1/20 0.41
HIF1A Q16665 1/20 0.41
CLK4 Q9HAZ1 1/20 0.41
KDM4E B2RXH2 1/20 0.41
CYP2C19 P33261 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29862626 1.00 CHEK2 (0.46) CHEK2CHEK1MAOBHTR6MKNK1
Hydrochloric Acid SCHEMBL29862870 0.99 CHEK2 (0.46) CHEK2CHEK1MAOBHTR6MKNK1
Hydrochloric Acid SCHEMBL23359980 0.99 CHEK2 (0.46) CHEK2CHEK1MAOBHTR6MKNK1
Hydrochloric Acid SCHEMBL29863199 0.99 CHEK2 (0.46) CHEK2CHEK1MAOBHTR6MKNK1
Hydrochloric Acid SCHEMBL23360234 0.99 CHEK2 (0.46) CHEK2CHEK1MAOBHTR6MKNK1
Hydrochloric Acid SCHEMBL23359983 0.99 CHEK2 (0.46) CHEK2CHEK1MAOBHTR6MKNK1
Hydrochloric Acid SCHEMBL23359856 0.92 CYP1A2 (0.46) HTR6MKNK1CYP1A2LMNACYP3A4
Hydrochloric Acid SCHEMBL29862635 0.92 CYP1A2 (0.46) HTR6MKNK1CYP1A2LMNACYP3A4
SCHEMBL29862805 0.85 HTR1A (0.54) CHEK2CHEK1MKNK1MKNK2AXL
Hydrochloric Acid SCHEMBL23360614 0.84 HTR1A (0.53) CHEK2CHEK1MAOBHTR6MKNK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114867719-A Pyrrolidine and piperidine compounds 柳韩洋行 2022-08-05 CN disclosed