SCHEMBL29866463

SCHEMBL29866463

CC(=O)Nc1cc([N+](=O)[O-])c(N(C)CCN(C)C)nc1OC(F)F

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 3/20 0.42
LMNA P02545 3/20 0.42
ALDH1A1 P00352 3/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
POLB P06746 2/20 0.42
GALR2 O43603 1/20 0.42
MITF O75030 1/20 0.42
HSP90AA1 P07900 1/20 0.42
HPGD P15428 1/20 0.42
XBP1 P17861 1/20 0.42
CCR6 P51684 1/20 0.42
MAPT P10636 3/20 0.39
KMT2A Q03164 5/20 0.36
HTT P42858 2/20 0.33
SLC9A1 P19634 1/20 0.33
CHEK1 O14757 1/20 0.32
DAPK3 O43293 1/20 0.32
PRKD3 O94806 1/20 0.32
MET P08581 1/20 0.32
PDGFRA P16234 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17490479 0.91 NPSR1 (0.40) NPSR1LMNAALDH1A1SMN1; SMN2POLB
SCHEMBL17490478 0.87 ALDH1A1 (0.42) NPSR1LMNAALDH1A1SMN1; SMN2POLB
Hydrochloric Acid SCHEMBL18979043 0.86 ALDH1A1 (0.41) NPSR1LMNAALDH1A1SMN1; SMN2POLB
SCHEMBL18978915 0.84 ALDH1A1 (0.40) NPSR1LMNAALDH1A1SMN1; SMN2POLB
SCHEMBL18978911 0.82 KDM4E (0.38) NPSR1LMNAALDH1A1SMN1; SMN2POLB
SCHEMBL18978910 0.82 KDM4E (0.38) NPSR1LMNAALDH1A1SMN1; SMN2POLB
SCHEMBL30459706 0.79 ALDH1A1 (0.43) NPSR1LMNAALDH1A1SMN1; SMN2POLB
SCHEMBL17490420 0.79 KDM4E (0.33) KDM4EGAA
SCHEMBL28359039 0.78 NPSR1 (0.45) NPSR1LMNAALDH1A1SMN1; SMN2POLB
SCHEMBL28359193 0.78 POLB (0.45) NPSR1LMNAALDH1A1SMN1; SMN2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110642838-B EGFR inhibitor and preparation and application thereof 江苏威凯尔医药科技有限公司 2022-08-09 CN disclosed