SCHEMBL29869

SCHEMBL29869

Clc1cc(Cl)n2nccc2n1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 2/20 1.00
KCNN3 Q9UGI6 14/20 0.51
KCNN1 Q92952 2/20 0.51
KCNN2 Q9H2S1 2/20 0.51
DPP4 P27487 2/20 0.35
CHEK1 O14757 1/20 0.32
CCNA2 P20248 1/20 0.32
CDK2 P24941 1/20 0.32
CCNA1 P78396 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29344715 0.80 PDE10A (0.67) PDE10AKCNN3KCNN1KCNN2
SCHEMBL30974 0.80 PDE10A (0.67) PDE10AKCNN3KCNN1KCNN2CHEK1
SCHEMBL659433 0.80 PDE10A (0.67) PDE10AKCNN3KCNN1KCNN2
SCHEMBL1018372 0.80 PDE10A (0.67) PDE10AKCNN3KCNN1KCNN2CHEK1
SCHEMBL13022182 0.80 PDE10A (0.67) PDE10AKCNN3KCNN1KCNN2DPP4
SCHEMBL1290450 0.80 PDE10A (0.67) PDE10AKCNN3KCNN1KCNN2DPP4
SCHEMBL312516 0.78 PDE10A (0.64) PDE10ACDK2
SCHEMBL12363999 0.76 PDE10A (0.61) PDE10AKCNN3KCNN1KCNN2
SCHEMBL1695626 0.76 PDE10A (0.61) PDE10AKCNN3KCNN1KCNN2
SCHEMBL14242902 0.76 PDE10A (0.61) PDE10AKCNN3KCNN1KCNN2DPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 456 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110016036-B Pyrazolo [1,5-a ] pyrimidine compound and preparation method and application thereof 辽宁大学 2022-06-03 CN claimed
CN-122094954-A Tricyclic quinolones and 1, 8-naphthyridin-2-one BCL6 difunctional degrading agents 2026-05-26 CN disclosed
CN-115943145-B Pyrazolopyrimidine compounds as ATR kinase inhibitors BEIJING TIDE PHARMACEUTICAL CO.,LTD. (CN) 2026-05-26 CN disclosed
US-12595263-B2 Pyrazolopyrimidine compound used as ATR kinase inhibitor BEIJING TIDE PHARMACEUTICAL CO., LTD. (CN) 2026-04-07 US disclosed
EP-4717312-A1 PYRAZOLO[1,5-A]PYRIMIDINE DERIVATIVES USEFUL AS A MEDICAMENT Perha Pharmaceuticals (FR) 2026-04-01 EP disclosed
EP-3778604-B1 LRRK2 INHIBITORS AND METHODS OF MAKING AND USING THE SAME DANA FARBER CANCER INST INC (US) 2026-01-07 EP disclosed
US-12479848-B2 Substituted fused heteroaromatic bicyclic compounds as kinase inhibitors and the use thereof Impact Therapeutics (Shanghai), Inc (CN) 2025-11-25 US disclosed
US-20250353852-A1 COMPOUNDS AND COMPOSITIONS THAT INHIBIT PIKFYVE KINETA INC (US) 2025-11-20 US disclosed
US-20250320219-A1 SUBSTITUTED FUSED HETEROAROMATIC BICYCLIC COMPOUNDS AS KINASE INHIBITORS AND THE USE THEREOF IMPACT THERAPEUTICS SHANGHAI INC (CN) 2025-10-16 US disclosed
US-20250270174-A1 CD73 COMPOUNDS GILEAD SCIENCES, INC. 2025-08-28 US disclosed
EP-1671962-A1 NOVEL FUSED HETEROCYCLIC COMPOUND AND USE THEREOF ONO PHARMACEUTICAL CO., LTD. (JP) 2006-06-21 EP disclosed
EP-1666468-A1 CRF ANTAGONISTS AND HETEROBICYCLIC COMPOUNDS ONO PHARMACEUTICAL CO., LTD. (JP) 2006-06-07 EP disclosed
EP-0628559-B1 Pyrimidine compounds and their use as pharmaceuticals BEIERSDORF LILLY GMBH (DE) 2002-04-03 EP disclosed
US-5602137-A Pyrimidine compounds and their use as pharmaceuticals BEIERSDORF-LILLY GMBH (DE) 1997-02-11 US disclosed
US-5602136-A Pyrimidine compounds and their use as pharmaceuticals BEIERSDORF-LILLY GMBH (DE) 1997-02-11 US disclosed
US-5571813-A Fused pyrimidine compounds and their use as pharmaceuticals BEIERSDORF-LILLY GMBH (DE) 1996-11-05 US disclosed
EP-0628559-A1 Pyrimidine compounds and their use as pharmaceuticals Beiersdorf-Lilly GmbH (DE) 1994-12-14 EP disclosed
US-4908056-A Herbicides E. I. DU PONT DE NEMOURS AND COMPANY (US) 1990-03-13 US disclosed
US-4838925-A HERBICIDES E. I. DU PONT DE NEMOURS AND COMPANY (US) 1989-06-13 US disclosed
EP-0244166-A2 Heterocyclic acetyl sulfonamides E.I. DU PONT DE NEMOURS AND COMPANY (US) 1987-11-04 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250353852-A1 COMPOUNDS AND COMPOSITIONS THAT INHIBIT PIKFYVE PIKFYVE, TARDBP, TDP1 PDE10A 2113/4885KCNN3 2131/4885KCNN1 2468/4885
US-20250320219-A1 SUBSTITUTED FUSED HETEROAROMATIC BICYCLIC COMPOUNDS AS KINASE INHIBITORS AND THE USE THEREOF ATR, CHEK1, CHEK2 PDE10A 3802/4885KCNN3 4247/4885KCNN1 4054/4885
US-20250270174-A1 CD73 COMPOUNDS ENTPD5, NT5E, ENTPD1 PDE10A 330/4885KCNN3 1294/4885KCNN1 1024/4885
US-12479848-B2 Substituted fused heteroaromatic bicyclic compounds as kinase inhibitors and the use thereof ATR, CHEK1, CHEK2 PDE10A 3837/4885KCNN3 4251/4885KCNN1 4041/4885
US-12595263-B2 Pyrazolopyrimidine compound used as ATR kinase inhibitor ATR, CHEK1, ATRIP PDE10A 3700/4885KCNN3 2925/4885KCNN1 2743/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.