SCHEMBL29883277

SCHEMBL29883277

C=CC(=O)N(Cc1cccnc1)c1ccc(Oc2ccccc2)c(C(F)(F)F)c1

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GSTO1 P78417 1/20 0.48
SUCNR1 Q9BXA5 1/20 0.42
GRM2 Q14416 6/20 0.42
PDK1 Q15118 4/20 0.42
NR1H4 Q96RI1 1/20 0.41
TP53 P04637 1/20 0.38
QPCT Q16769 1/20 0.38
CETP P11597 1/20 0.38
GAA P10253 1/20 0.38
TSHR P16473 1/20 0.38
MAPT P10636 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18763021 1.00 GSTO1 (0.48) GSTO1SUCNR1GRM2PDK1NR1H4
SCHEMBL21168598 0.88 CYP3A4 (0.46) SUCNR1GRM2PDK1NR1H4TP53
SCHEMBL18778620 0.86 GSTO1 (0.51) GSTO1GRM2TP53QPCTMAPT
SCHEMBL6728076 0.84 CYP3A4 (0.49) SUCNR1GRM2PDK1NR1H4TP53
SCHEMBL22866462 0.80 GRM2 (0.43) SUCNR1GRM2PDK1CETPMAPT
SCHEMBL6739000 0.78 GRM2 (0.56) GRM2GAA
SCHEMBL6736418 0.78 GRM2 (0.53) GRM2
SCHEMBL20857053 0.78 BCL2A1 (0.43) MAPT
SCHEMBL6734194 0.77 GRM2 (0.69) GRM2
SCHEMBL18763043 0.77 GSTO1 (0.50) GSTO1PDK1NR1H4GAATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4045050-A1 AN ACTIVITY-GUIDED MAP OF ELECTROPHILE-CYSTEINE INTERACTIONS IN PRIMARY HUMAN IMMUNE CELLS The Scripps Research Institute (US) 2022-08-24 EP disclosed