SCHEMBL29886232

SCHEMBL29886232

COc1cc(Cl)c(Cl)c(Cl)c1N1CCN(C(=O)OC(C)(C)C)[C@@H](C(=O)O)C1

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 8/20 0.42
NR1H3 Q13133 7/20 0.42
SUV39H2 Q9H5I1 3/20 0.41
ALDH1A1 P00352 1/20 0.37
MCL1 Q07820 1/20 0.36
OPRK1 P41145 1/20 0.35
ALK Q9UM73 2/20 0.35
CCR1 P32246 2/20 0.35
HSD17B10 Q99714 1/20 0.35
LMNA P02545 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23216745 1.00 NR1H2 (0.42) NR1H2NR1H3SUV39H2ALDH1A1MCL1
SCHEMBL29768486 1.00 NR1H2 (0.42) NR1H2NR1H3SUV39H2ALDH1A1MCL1
SCHEMBL29768375 0.91 NR1H2 (0.41) NR1H2NR1H3SUV39H2ALDH1A1ALK
SCHEMBL23239752 0.91 NR1H2 (0.52) NR1H2NR1H3SUV39H2ALDH1A1ALK
SCHEMBL23239747 0.91 NR1H2 (0.41) NR1H2NR1H3SUV39H2ALDH1A1ALK
SCHEMBL23216453 0.88 NR1H2 (0.42) NR1H2NR1H3SUV39H2ALDH1A1MCL1
SCHEMBL29886243 0.88 NR1H2 (0.42) NR1H2NR1H3SUV39H2ALDH1A1MCL1
SCHEMBL29768376 0.88 NR1H2 (0.42) NR1H2NR1H3SUV39H2ALDH1A1MCL1
SCHEMBL23215030 0.87 ALDH1A1 (0.36) ALDH1A1CCR1HSD17B10
SCHEMBL23239713 0.78 NR1H2 (0.41) NR1H2NR1H3SUV39H2ALDH1A1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4041407-A1 ARYL HETEROCYCLIC COMPOUNDS AS KV1.3 POTASSIUM SHAKER CHANNEL BLOCKERS D.E. Shaw Research, LLC (US) 2022-08-17 EP disclosed