SCHEMBL29890958

SCHEMBL29890958

CN1CCN(c2ccc([N+](=O)[O-])cc2Nc2ncnc(Cl)c2[N+](=O)[O-])CC1

nearest known ligand 0.80

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
WDR5 P61964 19/20 0.80
KMT2A Q03164 11/20 0.80
ALDH1A1 P00352 1/20 0.52
CYP2D6 P10635 1/20 0.52
GAA P10253 1/20 0.50
EIF2AK2 P19525 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24429937 1.00 WDR5 (0.80) WDR5KMT2AALDH1A1CYP2D6GAA
SCHEMBL24429939 0.90 WDR5 (0.80) WDR5KMT2AALDH1A1CYP2D6GAA
SCHEMBL29890970 0.90 WDR5 (0.80) WDR5KMT2AALDH1A1CYP2D6GAA
SCHEMBL29544609 0.89 WDR5 (1.00) WDR5KMT2A
SCHEMBL24429879 0.89 WDR5 (1.00) WDR5KMT2A
SCHEMBL24429921 0.87 WDR5 (0.76) WDR5KMT2AALDH1A1CYP2D6GAA
SCHEMBL29891312 0.87 WDR5 (0.79) WDR5KMT2AALDH1A1CYP2D6GAA
SCHEMBL24429882 0.87 WDR5 (0.79) WDR5KMT2AALDH1A1CYP2D6GAA
SCHEMBL29891004 0.87 WDR5 (0.76) WDR5KMT2AALDH1A1CYP2D6GAA
SCHEMBL24429900 0.86 WDR5 (0.75) WDR5KMT2AALDH1A1CYP2D6GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109734674-B Aniline WDR5 protein-protein interaction inhibitor and preparation method and application thereof 中国药科大学 2022-08-26 CN disclosed