SCHEMBL29891722

SCHEMBL29891722

Cn1c(=O)c(Br)cc2ccccc21

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DAO P14920 1/20 0.62
CA12 O43570 2/20 0.50
CA9 Q16790 2/20 0.50
BRD4 O60885 1/20 0.50
BRPF1 P55201 1/20 0.50
KAT2B Q92831 1/20 0.50
BRD9 Q9H8M2 1/20 0.50
MCL1 Q07820 1/20 0.49
KMT2A Q03164 5/20 0.47
AHR P35869 3/20 0.47
DDB1 Q16531 1/20 0.47
CRBN Q96SW2 1/20 0.47
GAA P10253 2/20 0.44
PKM P14618 1/20 0.44
CASP1 P29466 1/20 0.44
GALK1 P51570 1/20 0.44
BLM P54132 1/20 0.44
CASP7 P55210 1/20 0.44
HSD17B10 Q99714 1/20 0.44
SAE1 Q9UBE0 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1421868 1.00 DAO (0.62) DAOCA12CA9BRD4BRPF1
SCHEMBL31426215 0.78 DAO (0.65) DAOCA12CA9BRD4BRPF1
SCHEMBL715895 0.78 DAO (0.65) DAOCA12CA9BRD4BRPF1
SCHEMBL11479451 0.78 DAO (0.42) DAOCA12CA9BRD4BRPF1
SCHEMBL31039545 0.77 DAO (0.62) DAOCA12CA9BRD4BRPF1
SCHEMBL30349848 0.77 DAO (0.62) DAOCA12CA9BRD4BRPF1
SCHEMBL8538250 0.77 DAO (0.62) DAOCA12CA9BRD4BRPF1
SCHEMBL10677691 0.77 KDM4E (0.52) DAOMCL1KMT2AAHRDDB1
SCHEMBL21955107 0.77 DAO (0.62) DAOCA12CA9BRD4BRPF1
SCHEMBL28165616 0.77 DAO (0.62) DAOCA12CA9BRD4BRPF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4548972-A2 (2S)-N-[(1S)-1-CYANO-2-PHENYLETHYL]-1,4-OXAZEPANE-2-CARBOXAMIDES AS DIPEPTIDYL PEPTIDASE I INHIBITORS AstraZeneca AB (SE) 2025-05-07 EP disclosed
CN-119462635-A Quinoline derivatives as alpha 4 beta 7 integrin inhibitors 吉利德科学公司 2025-02-18 CN disclosed
CN-112969687-B Quinoline derivatives as a4 b 7 integrin inhibitors 吉利德科学公司 2024-08-23 CN disclosed
CN-112969700-B Imidazopyridine derivatives as alpha 4 beta 7 integrin inhibitors 吉利德科学公司 2024-08-20 CN disclosed
CN-112996786-B Compounds for inhibiting alpha 4 beta 7 integrin 吉利德科学公司 2024-08-20 CN disclosed
CN-112969504-B Compounds for inhibiting alpha 4 beta 7 integrin 吉利德科学公司 2024-04-09 CN disclosed
CN-115003665-A Substituted aminoquinolones as immunoactive DGK alpha inhibitors 拜耳公司 2022-09-02 CN disclosed