SCHEMBL2990185

SCHEMBL2990185

CC(C)(C)OC(=O)Cc1ccc(Oc2ccc(C(=O)NC(Cl)Cc3ccc(Cl)cc3)c(F)c2)c(C#N)c1

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
EZH2 Q15910 1/20 0.38
PLA2G7 Q13093 4/20 0.37
MAOA P21397 1/20 0.37
MAOB P27338 1/20 0.37
PTGDR2 Q9Y5Y4 2/20 0.37
PTGDR Q13258 1/20 0.35
ACACB O00763 2/20 0.35
CTSB P07858 1/20 0.35
LMNA P02545 1/20 0.35
TRPA1 O75762 1/20 0.35
S1PR3 Q99500 5/20 0.34
P2RX7 Q99572 1/20 0.34
SLC22A12 Q96S37 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2986773 0.89 PTGDR2 (0.40) EZH2PLA2G7MAOAMAOBPTGDR2
SCHEMBL2990179 0.81 PTGDR2 (0.43) EZH2PLA2G7PTGDR2PTGDRSLC22A12
SCHEMBL2982722 0.76 PTGDR2 (0.51) PLA2G7PTGDR2PTGDRS1PR3
SCHEMBL2983525 0.75 PTGDR2 (0.47) PTGDR2S1PR3
SCHEMBL2986695 0.74 PTGDR2 (0.54) PTGDR2PTGDR
SCHEMBL2984362 0.71 MAPK14 (0.40) PLA2G7LMNA
SCHEMBL2988579 0.71 CACNA1H (0.45) PLA2G7TRPA1
SCHEMBL2990233 0.71 LPAR1 (0.49) PLA2G7PTGDR2
SCHEMBL2986772 0.70 PTGDR2 (0.48) EZH2PTGDR2PTGDR
SCHEMBL2986645 0.69 PLA2G7 (0.48) PLA2G7PTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8492437-B2 4-substituted phenoxyphenylacetic acid derivatives ARRAY BIOPHARMA INC. (US) 2013-07-23 US disclosed
EP-2057115-B9 4-SUBSTITUTED PHENOXYPHENYLACETIC ACID DERIVATIVES ARRAY BIOPHARMA INC (US) 2012-12-26 EP disclosed
EP-2057115-B1 4-SUBSTITUTED PHENOXYPHENYLACETIC ACID DERIVATIVES ARRAY BIOPHARMA INC (US) 2012-10-03 EP disclosed
US-20120202854-A1 4-SUBSTITUTED PHENOXYPHENYLACETIC ACID DERIVATIVES ARRAY BIOPHARMA INC. (US) 2012-08-09 US disclosed
US-8183289-B2 4-substituted phenoxyphenylacetic acid derivatives ARRAY BIOPHARMA INC. (US) 2012-05-22 US disclosed
US-20100173955-A1 4-SUBSTITUTED PHENOXYPHENYLACETIC ACID DERIVATIVES ARRAY BIOPHARMA INC. (US) 2010-07-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100173955-A1 4-SUBSTITUTED PHENOXYPHENYLACETIC ACID DERIVATIVES CD22, HRH2, CD74 EZH2 3601/4885PLA2G7 1735/4885MAOA 2010/4885
US-20120202854-A1 4-SUBSTITUTED PHENOXYPHENYLACETIC ACID DERIVATIVES CD22, HRH2, CD74 EZH2 3601/4885PLA2G7 1735/4885MAOA 2010/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.