SCHEMBL29907491

SCHEMBL29907491

CN(C)c1ccnc(C#N)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM5 P08912 1/20 0.46
CHKA P35790 1/20 0.46
ALDH1A1 P00352 4/20 0.46
KDM4E B2RXH2 1/20 0.46
XDH P47989 1/20 0.40
ABCG2 Q9UNQ0 1/20 0.40
MYC P01106 1/20 0.39
HPGD P15428 3/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
RAB9A P51151 2/20 0.39
HTT P42858 2/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
JAK2 O60674 1/20 0.39
JAK1 P23458 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22551997 1.00 CHRM5 (0.46) CHRM5CHKAALDH1A1KDM4EXDH
SCHEMBL2222144 0.93 ALDH1A1 (0.41) CHRM5CHKAALDH1A1KDM4EXDH
SCHEMBL2222139 0.90 ALDH1A1 (0.42) CHRM5CHKAALDH1A1KDM4EXDH
SCHEMBL19462352 0.76 MAPT (0.38) ALDH1A1KDM4EXDHABCG2MYC
SCHEMBL2192891 0.76 GRM5 (0.45) XDHABCG2
SCHEMBL91455 0.72
SCHEMBL30078627 0.72
SCHEMBL3354091 0.72 SRC (0.39) ALDH1A1KDM4EMYCCYP1A2CYP3A4
SCHEMBL196641 0.72 ALDH1A1 (0.53) CHRM5CHKAALDH1A1KDM4ESMN1; SMN2
SCHEMBL31133396 0.72 MYC (0.62) XDHABCG2MYCNPY5R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115181092-B Pyrazine compounds and uses thereof 迪哲(江苏)医药股份有限公司 2024-05-03 CN disclosed
CN-115181092-A Pyrazine compounds and uses thereof 迪哲(江苏)医药股份有限公司 2022-10-14 CN disclosed
CN-112279837-B Pyrazine compounds and uses thereof 迪哲(江苏)医药股份有限公司 2022-08-09 CN disclosed