SCHEMBL29907684

SCHEMBL29907684

COC(=O)c1nc(Cl)c(-c2ccc(F)cc2)nc1N

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.51
PKM P14618 5/20 0.45
KDM4E B2RXH2 5/20 0.45
ALDH1A1 P00352 3/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
L3MBTL1 Q9Y468 2/20 0.45
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
CASP3 P42574 1/20 0.44
SENP8 Q96LD8 1/20 0.44
SENP7 Q9BQF6 1/20 0.44
SENP6 Q9GZR1 1/20 0.44
MAPT P10636 3/20 0.43
IKBKB O14920 1/20 0.43
RCE1 Q9Y256 1/20 0.42
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA9 Q16790 1/20 0.42
ADORA2A P29274 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21730350 1.00 LMNA (0.51) LMNAPKMKDM4EALDH1A1SMN1; SMN2
SCHEMBL22551809 0.86 KDM4E (0.46) LMNAPKMKDM4EALDH1A1SMN1; SMN2
SCHEMBL29907784 0.86 KDM4E (0.46) LMNAPKMKDM4EALDH1A1SMN1; SMN2
SCHEMBL22551772 0.86 KDM4E (0.40) LMNAPKMKDM4EALDH1A1SMN1; SMN2
SCHEMBL5425548 0.86 SMN1; SMN2 (0.52) PKMKDM4EALDH1A1SMN1; SMN2L3MBTL1
SCHEMBL21730335 0.85 ATR (0.41) PKMKDM4EALDH1A1SMN1; SMN2L3MBTL1
SCHEMBL22579104 0.85 MAPT (0.40) LMNAPKMKDM4EALDH1A1L3MBTL1
SCHEMBL21722384 0.84 PLAU (0.43) LMNAKDM4EALDH1A1IKBKBADORA2A
SCHEMBL21730378 0.84 TDP1 (0.44) ADORA2APLAUDHODH
SCHEMBL29907506 0.84 TDP1 (0.44) ADORA2APLAUDHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115181092-B Pyrazine compounds and uses thereof 迪哲(江苏)医药股份有限公司 2024-05-03 CN disclosed
CN-115181092-A Pyrazine compounds and uses thereof 迪哲(江苏)医药股份有限公司 2022-10-14 CN disclosed
CN-112279837-B Pyrazine compounds and uses thereof 迪哲(江苏)医药股份有限公司 2022-08-09 CN disclosed